ImpiloAmalungiselelo

"Kofetamin": yokusetshenziswa, analogs, isithombe, ukubuyekezwa

Migraine sibizwa ngokuthi isifo esithinta izinzwa ukuthi ngokuhlaselwa njalo noma ngezikhathi ezithile obedlulele okunzima ubuhlungu, okuyinto eyenzeka ngo-nengxenye eyodwa ekhanda. isiguli okunjalo ongakaphathelani bathola ukulimala okunzima, unhlangothi noma ebuchosheni. Imvelo onesigqi futhi ukushuba ubuhlungu ukuchaza khona izilonda semithambo, kanti isiguli akuyona voltage ngokweqile.

Kufanele kuphawulwe ukuthi ubuhlungu bekhanda migraine awahlobene nokwehla abukhali noma ukwanda wegazi, ukuquleka, ingcindezi intracranial noma ukufiphala kwamehlo.

ochwepheshe abaningi batusa usebenzisa imithi "Kofetamin" ukwelapha isimo. Yokusetshenziswa, izidakamizwa isithombe, ukubuyekezwa ngakho, amathuluzi ezifanayo futhi izici tibalwe lapha ngentasi.

Ukwakheka izidakamizwa futhi ifomu ikhishwe futhi emaphaketheni

Yini ifomu owenza izidakamizwa "Kofetamin"? Yokusetshenziswa, izimpendulo ezibonisa ukuthi lesi sakhiwo itholakale ukudayiselwa ngesimo amaphilisi. Bahlanganisa izithako ezifana ergotamine tartrate, amazambane isitashi, stearic acid, talc, i-caffeine, glucose kanye noshukela.

Ukudayiswa kwezidakamizwa elinikelwe amabhamuza.

izici Pharmacodynamic imithi

Ithebhulethi emangalisayo "Kofetamin"? Yokusetshenziswa busikisela ukuthi leli kuhlanganiswe izindlela, okuyinto ngenxa izakhiwo izithako kwengoma.

Caffeine kusiza ukushukuma vasomotor futhi izikhungo zokuphefumula, kodwa futhi sithuthukisa excitation we- cortex. Ngaphezu kwalokho, lokhu izidakamizwa has a action cardiotonic. It kancane kwandisa umfutho wegazi futhi kwandisa izinga emishinini yokuphefumula nokushaya kwenhliziyo. Caffeine futhi kunciphisa ukozela, kuvusa umsebenzi locomotor, aqede ukukhathala, kuthuthukisa impilo jikelele.

Umonakalo obangelwa nobude le ngxenye kuncike isimo somuntu, ezifana isimiso sezinzwa futhi umsebenzi wonke umzimba.

Ngemithamo emincane caffeine kunomphumela Ugqozi, nokuningi - umphumela ezicindezelayo phezu CNS.

Kepha ergotamine, ke kunomphumela vasoconstrictor.

izici kinetic

Lapho ukumuncwa izimali ngokuthi "Kofetamin"? Yokusetshenziswa busikisela ukuthi leli umuthi ngempela okuhle kanye kakhulu ngokushesha ugxile kusukela amathumbu. Ergotamine 98% eboshiwe plasma amaphrotheni, i-caffeine - by 35%.

Ubuningi esiphezulu izidakamizwa egazini waphawula ngemva kwamahora angu-2 emva nokuphathwa tablet. Ingxenye esemqoka caffeine is oxidized bese demethylated, bese siboniswa umchamo.

umzimba Ergotamine esibindini esebumba nemikhiqizo asebenzayo.

Lokhu ukulungiselela isuselwe ogxile e Bile amahora amahlanu.

Izinkomba ukuthola amaphilisi okwelapha

Kungakhathaliseki ukuthi uyazi inhloso angabelwa yokukhalaza "Kofetamin"? Imiyalelo, ukubuyekezwa ukubika ukuthi lo muthi siyasebenza kakhulu ngefomu vazoparaliticheskoy migraine, hypotension, kanye izilonda senhliziyo, izifo kanye ebuhlungu isimiso sezinzwa esiyinhloko, isetshenziswa yokunciphisa izingcindezi intracranial.

Uvala izidakamizwa ukusetshenziswa

Lapho hhayi prescribers "Kofetamin"? Ukufundiswa (izidakamizwa analogue ezibalwe ngezansi) ibika ukuthi ithuluzi asivunyelwe ukuthatha ngesikhathi sensitivity high emuthini, kanye ngesikhathi sokukhulelwa futhi ngesikhathi lactation.

Ngokunakekela ukuthi nomuthi isetshenziswa uma eshiwo iziyaluyalu ubuthongo, umfutho ophakeme wegazi, izifo semithambo futhi inhliziyo (isb, angina, isifo sokuqina kwemithambo yegazi, tachycardia paroxysmal, isilethikusebenza, neuropathy isifo semithambo), ukufiphala kwamehlo nokukhathazeka netwetwe neziyaluyalu, izinso, isibindi, agoraphobia kanti lapho esekhulile.

Izidakamizwa "Kofetamin": yokusetshenziswa

Analogue lomutsi Kufanele umise udokotela kuphela. Lokhu kungenxa yokuthi bangase babe izinhlobo ezihlukene kakhulu ukwakhiwa kanye nezindlela zokusebenzisa.

Lo muthi kufanele busetshenziswe phakathi zekhanda ezinamandla. Kulokhu, iqondiswa e isamba 1-2 amaphilisi kabili ngelanga. Ngemva kwalokho, izinsuku ezimbalwa imithi ukuthatha 1 tablet kaningi efanayo.

Ungalokothi idlule esiphezulu umthamo owodwa elilingana amaphilisi 2 nsuku zonke futhi ilingana 4.

Kufanele kuphawulwe ukuthi akufanele uthathe isidakamizwa olucutshungulwayo isikhathi eside. Ngemva kwesonto ukusetshenziswa kwezidakamizwa kuyadingeka ukwenza ikhefu izinsuku 4.

side effects

Mayelana yimuphi imiphumela engemihle engase baqaphe ngaphambi uthatha "Kofetamin" ithebhulethi? Ukufundiswa zomuthi uthi kungabangela ukusabela ezilandelayo:

  • Cardialgia, isiyezi, hypertonia, excitation;
  • tachycardia, ikhanda elibuhlungu, ukukhathazeka, ukulunywa, ukukhathazeka, ukundindizela, ikhaliphe anda, isicanucanu, ukuqwasha;
  • uhudo, amajaqamba, ukuhlanza, paresthesia e emikhawulweni, ukuvuvukala.

Uma imithi yokwelapha eside zingase ukuthuthukisa myalgias, ukuphazamiseka jikelele sezinzwa ezingalweni nasemilenzeni ephansi, noma ukuba buthakathaka.

Overdose nezidakamizwa ekuxhumaneni

Yiziphi izimpawu ukweqisa izidakamizwa zenzeka ngemithamo lapho ephakeme zomuthi ngokuthi "Kofetamin"? Imiyalelo isicelo uthi kulesi simo manifest nesineke: ukozela, isicanucanu, ukucobeka, ukuhlanza, ukuba ndikindiki eminweni wemikhawulo engenhla nengezansi, stupor, futhi sokuwa futhi equlekile. Ukuqeda izenzakalo ezinjalo ukuqhuba lavage esiswini. Futhi, isiguli isebenze namalahle.

Lokhu imithi kwandisa imiphumela izidakamizwa, ezibandakanya ergot alkaloids ne-caffeine. Uma is kuhlangene barbiturates futhi anticonvulsants kwandisa imvume caffeine kanye ngesivinini umzimba walo.

I-nicotine ikhuthaza ukususwa okusheshayo zomuthi, futhi CNS evuselela - excitability ngokweqile.

nomuthi Okubukwe kunciphisa umphumela izidakamizwa okuyiluthayo, analgesics kwezidakamizwa, futhi kwandisa ukumuncwa futhi ubuthi glycosides zenhliziyo analgesics non-kwezidakamizwa.

Co-ekuphathweni caffeine-beta-blocker ngokuvamile kuholela ukucindezelwa mutual imiphumela yabo zokwelapha futhi bronchodilators adrenergic - ukuze sikhuthaze isimiso sezinzwa nezinye okufakiwe ukusabela anobuthi.

Phawula futhi ukuthi isithako esebenzayo zomuthi kunganciphisa imvume theophylline nezinye xanthines.

Umsebenzi vasoconstrictor zomuthi ukwanda beta-blocker, i-alpha-adrenostimulyatorov, nicotine kanye serotonin agonists.

I ubuthi ergotamine ukwanda macrolides.

Izindleko imithi izidakamizwa futhi efanayo

Thenga le-ejenti e isamba amaphilisi 10 unga ruble 100-150. Uma kudingeka, kungase kuthathelwe indawo izidakamizwa ezifanayo njenge "Kofergot", "Ergofeyn", "Nomigren", "Ergoffin". Kodwa kungakenzeki lokho, qiniseka ukuthi uxhumane nodokotela wakho.

Izibuyekezo ochwepheshe kanye neziguli

Manje unombono kanjani imithi "Kofetamin". Ukusetshenziswa salo mhlahlandlela kusho njengoba kuchaziwe ngenhla. Izimpendulo ngaye lingama omuhle. Labo abantu abasebenzisa le ndlela yokuxhumana, bethi siwumsebenzi ngempumelelo yokulwa migraine ezinzima. a Amalungiselelo anjalo iphumelela kakhulu kunokuba wena nezinye izidakamizwa ezibiza kakhulu,. Abathengi ukubika ukuthi kwanele ukuthatha amaphilisi amabili ngosuku. Isikali enjalo ngokushesha aqede ubuhlungu. Nakuba ngezinye izikhathi ukungakhululeki ukuhlala ngisho nangemva izidakamizwa abaphathi. Kodwa kulokhu kungukuthi libizwa.

La maqembu engakhi ithuluzi zihlanganisa inani elikhulu ohlangothini ukusabela ukuba senziwe ngemuva reception yayo.

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