ImpiloAmalungiselelo

'Betalok' yokusetshenziswa

"Betalok" imfundo manual uchaza njengoba izidakamizwa okuqondene kwemithi iqembu beta1-adrenoceptor abantu abamelene nani. The main isithako zomuthi kuyinto metoprolol tartrate. It ikhiqizwa yizimboni ngesimo amaphilisi enesisindo angu 100, ingalendlela e amabhodlela epulasitiki yizicucu 100 ngamunye.

"Metoprolol" anezakhi kwemithi, esekelwe ikhono zomuthi ukunikeza antihypertensive futhi isenzo eqeda anginal. Umuthi ngempumelelo ekunciphiseni izinga lokushaya kwenhliziyo, contractility esivimba amanzi futhi excitability, lwenza deceleration izinqubo AV-conduction. Ukulungiselela "Betalok" imfundo manual uchaza njengenhlangano aid nokuncipha ivolumu zenhliziyo umoyampilo sokudliwa myocardium. "Metoprolol" uyakwazi ukunciphisa imithelela catecholamines at inkanuko umthelela wabo inhliziyo yesiguli ngesikhathi ukucindezeleka psycho-ngokomzimba. Umuthi kunomphumela hypotensive, eliletha ukuthula ngemva kwamasonto amabili yokwelashwa. "Metoprolol" libonisa kusebenta eyanele ekwelapheni a spectrum ebanzi izifo zenhliziyo, phakathi ezingasetshenziswa kuqashelwe isilethikusebenza, yenhliziyo Umthambo isifo, arrhythmias ezinhlobo ezehlukene, sisebenza-ejenti prophylactic ukuvimbela Ukuphinda ukuhlaselwa isifo senhliziyo.

izakhiwo Pharmacokinetic "Betalok" imiyalelo izidakamizwa ukusetshenziswa abachazwa ngale ndlela. Lapho ethola kakhulu zonke izidakamizwa ngesikhathi esifushane futhi ugxile kusukela ipheshana emathunjini, emakamu yayo esiphezulu ku-plasma litholakala ngaphakathi ihora elilodwa noma amabili. Umuthi ungakwazi ngokushesha akheka esibindini, metabolites ngaleyo ndlela ekhiqizwa babe cishe akukho msebenzi noma ngokuphikisana emizimbeni umzimba. Ingxenye-ukuphila yezingxenye umuthi amahora cishe emithathu kuya kwemine, futhi cishe akashintshi phakathi naso sonke isikhathi sokwelashwa. Excretion of metoprolol ikhiqizwa izinso - ezingaphezu kuka-95% umthamo lomcebo, lapho abangeqile kwabathathu amaphesenti is excreted zinjalo.

"Betalok" Umhlahlandlela incoma ukuthi ezimeni lezi zifo ezilandelayo: ukwelapha umfutho ophakeme wegazi, njenge-agent zokwelapha isetshenziswa ukuvimbela imivimbo. Umuthi kuboniswe amacala arrhythmias inhliziyo, kanye nokuvinjelwa yesibili kwakudingeka hlupheka uhlelo cardio-semithambo.

I umthamo lwemithi yebhukwana izidakamizwa "Betalok" imfundo incoma ukuthi ufake lolu. Umthamo isilinganiso izidakamizwa kabili ngosuku ngesikhathi yokwamukela angu 100 ngosuku. Kwezinye izimo, le mfundo sinika kungenzeka ukwenyuka kancane umthamo kabili. Uma izidakamizwa isetshenziswa ngemithambo yegazi, umthamo owodwa kuhluka 2 kuya 5 mg. Uma kuleli cala is hhayi izuzwe siletha imiphumela efiselekayo, ukulungiswa ingasatshenziswa ngokuphindaphindiwe emva kwemizuzu 5.

Isimiso Isikali kumele licubungule ukuthi isicelo umthamo esiphezulu umuthi 400 mg ngosuku.

Lapho ethola amaphilisi "Betalok" kungase kubangele imiphumela emibi evela izinhlelo ezihlukahlukene zomzimba. hlu yabo enemininingwane nencazelo izimpawu kunikezwe imiyalo ukusetshenziswa kwezidakamizwa.

Izimo ukuthola imithi ehlukene ngokwendlela uhlobo nohlobo ukugeleza ukuvinjelwa conductivity zenhliziyo, hypotension, ukushaqeka cardiogenic kanye nezinye izifo. Contraindicated reception uma isiguli hypersensitivity kuya izingxenye zalo. Musa thatha izidakamizwa ngenkathi bekhulelwe nangenkathi bencelisa.

Ngokucophelela okukhulu kufanele basondela ukuze ukusetshenziswa kwezidakamizwa iziguli kanye COPD,

isifo sikashukela, isifo Raynaud sika.

Imisa imithi Kunconywa kancane kancane, le nqubo kumele kutsatse okungenani izinsuku eziyishumi.

Umuthi enezinto eziningi izindlela ezikhethekile isinyathelo, ngokuhlanganisa ke neminye imithi. Lokhu ukwaziswa okuningiliziwe itholakala yokusetshenziswa.

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