ImpiloAmalungiselelo

Yokusetshenziswa "klopiksol" incazelo izidakamizwa, ukubuyekezwa

Kuyini lokhu izidakamizwa ngokuthi "klopiksol"? Umthengi ukubuyekezwa kanye izici zalesi izidakamizwa ezocatshangelwa mathiriyeli lo sihloko.

Ifomu sokulungiselela, ukubunjwa, incazelo, emaphaketheni

Kulaba izimali babe amafomu ahlukene ukukhululwa. Sethula kubo manje.

1. "klopiksol" - amaphilisi ayilutho pink, umbala pink onsundu ngokubomvu futhi iba nsundu ngokubomvu (2 mg, 10 mg kanye 25 mg, ngokulandelana). Ziyakwazi ukuma isiyingi futhi we-lenticular wangakwesokunxele, futhi ifilimu enamathela.

Isici esebenzayo ye thuluzi zuclopenthixol dihydrochloride. Futhi, siqukethe 85% glycerol, amazambane isitashi, copovidone, monohydrate lactose, microcrystalline cellulose, talc, magnesium stearate, uwoyela, hydrogenated ocolisekileyo.

Ngo ukudayiswa wayebheka izidakamizwa iza nezipakupaku futhi mabhokisi amakhadibhodi.

2. Isixazululo namafutha / m "klopiksol". Izibuyekezo bathi leli thuluzi okuthengiswa ampoules ezenziwe ngengilazi kungekho nto enemibala emihle. Isixazululo ngokwayo has a umbala aphuzi futhi obala. He is ngokuphelele khulula kusukela ezinhlayiyeni.

Isici esebenzayo lokhu imithi decanoate zuclopenthixol. Futhi liqukethe triglyceride.

Kwemithi isenzo "klopiksol"

nomuthi Okubukwe kuyinto esuselwe thioxanthene - a neuroleptic. Anakho imiphumela ethize inhibitory futhi antipsychotic. Ngaphezu kwalokho, ithuluzi ibonisa umphumela okulalisayo.

A ekuphathweni eyodwa izidakamizwa kunomthelela ekubeni buthakathaka okusheshayo izimpawu ngengqondo. izakhiwo sine zomuthi wabonakaliswa ngemva kwamahora angu-2, kanye nomphumela walo jikelele luthatha izinsuku 3.

izici Kinetic ekulungisweni

Ngokusho kochwepheshe, umjovo lokhu isixazululo kungcono ukuba afeze ngqi (njalo emavikini 4).

Ukulandela ekuphathweni temlomo, isiqongo izidakamizwa lokuhlushwa izuzwe emva 4 h. Zuclopenthixol bioavailability imayelana 44%.

Ukulandela ekuphathweni esicutshini into eyisisekelo yaleli ukulungiselela is phansi cleavage enzymatic. Lokhu kukhipha acetic acid kanye zuclopenthixol asebenzayo. Uphiko wokugcina okuncane excreted ku ubisi lwebele futhi lingena isithiyo esinomhlapho.

Lapho ethola nemithi isiwombe ukuphila isikhathi salo amahora angu-20. Libonisa ngokuyinhloko indle futhi kancane - ne umchamo.

Izinkomba ukusetshenziswa

Kwezinye izimo, umuthi ezinqunyiwe iziguli kubhekwe? Elikushoyo ngakho yokusetshenziswa? "Klopiksol" siboniswa:

  • bayasangana oyingozi futhi ezingalapheki nezinye izifo zengqondo, kuhlanganise nalezo okuyize ezihilela (Paranoid), ukusangana neziyaluyalu ekucabangeni;
  • isimo ukuyaluza, ubutha, ukukhathazeka (aphakeme), ulaka;
  • retardation engqondo, okuyinto kuhlangene ukuyaluza, ukuyaluza (lengqondo) nakwezinye iziyaluyalu ekuziphatheni;
  • mania ka sengqondo ukwenama-bacindezeleke;
  • komqondo senile, disorientation, ukuziphatha kahle, imibono paranoid futhi ukudideka.

Uvala izidakamizwa ukusetshenziswa

Lapho kufanele ungasebenzisi neuroleptic ukubika? Elikushoyo ngakho yokusetshenziswa? "Klopiksol" is contraindicated ku:

  • ukudakwa acute nge barbiturates;
  • acute utshwala ukudakwa nemvelo;
  • acute ukudakwa analgesics (opioid).

Kufanele kuphawulwe ukuthi kusho umphenyi antipsychotic alisetshenziswa isimo comatose.

Yokusetshenziswa

"Klopiksol" amaphilisi athathwa ngomlomo. Umthamo lokhu izidakamizwa kuyakhethwa ngamunye kuncike isimo lesiguli. Ekuqaleni yokwelapha izidakamizwa iqondiswa ngemithamo ongaphakeme, bese ngokushesha anda ukuze umphumela yabo emtholampilo.

Lapho uzwakalise nokulinganisela iziyaluyalu ingqondo umthamo kokuqala "klopiksol" 20 mg ngosuku. Uma kudingeka, kungase senyukela mg 20.

Ngo-acute isiqephu bayasangana nezinye izifo zengqondo, nemvelo acute, mania futhi ezinzima imithi ukuyaluza umthamo kuyinto 10-50 mg ngosuku.

Lapho ezingamahlalakhona uthi ingqondo imvelo, kanye bayasangana nezinye kwengqondo Isikali kubhekwe asekelayo izindlela 20-40 mg ngosuku.

Lapho ukuyaluza kubantu abanegciwane retardation engqondo umthamo kuyinto 6-20 mg ngosuku. Uma kudingeka, kungase senyukela 25-40 mg ngosuku.

Lapho iziyaluyalu senile ukuyaluza nokudideka lokhu izidakamizwa iqondiswa e umthamo 2-6 mg ngosuku. Uma kudingeka, lemali ebekiwe zomuthi luyanda 10-20 mg ngosuku.

Sokuphuzisa isixazululo uwoyela

okumele ngiyifake kanjani ikhambi uwoyela? Yini lokhu ekutshela imfundo manual? "Klopiksol" yaphathwa ngendlela ejulile / m umjovo owenziwa kule ndawo gluteal.

Inani watusa umjovo anjalo kufanele kube 1-3 ml. Uma kudingeka, okuphindaphindiwe imijovo wenza ngezikhawu izinsuku 3. Ezinye ezengeziwe iziguli imijovo Bamiswa ngemva kosuku noma ezimbili.

sequela engadingeki

Yini ukusabela okungekuhle kubangela izidakamizwa "klopiksol"? Imiphumela engemihle yalesi izidakamizwa kuvamile. Lezi zihlanganisa lokhu okulandelayo:

  • nokugcinwa urinary, ccomodation;
  • izimpawu extrapyramidal (esigabeni sokuqala yokwelapha), ukozela;
  • tachycardia, isiyezi, hypotension orthostatic ;
  • dyskinesia tardive (ukwelashwa nokunwetshiwe);
  • ukuqunjelwa, nomlomo owomile, izinguquko lezivakashi e umsebenzi ukuhlolwa isibindi.

amacala ukweqisa izidakamizwa

Nge ukweqisa izidakamizwa izimali, okulandelayo zimpawu: ikhoma, ukozela, Ukudlikizela, disorder extrapyramidal, ukushaqeka, hypotension, hypo- noma komzimba okukhulu.

Ukuqeda nesineke ezifana izenzakalo sagezwa esiswini futhi unike sorbents. Futhi, nokwelapha ongisekelayo lingaze.

izidakamizwa ekuhlanganyeleni

Ukulungiselela "klopiksol" (10 mg) sithuthukisa umphumela okulalisayo utshwala, barbiturates nezinye izidakamizwa okuyinto nomphumela inhibitory phezu CNS.

Lesi sidakamizwa akufanele kuhlangene guanethidine nezidakamizwa ne zinemiphumela efanayo ngenxa kungenzeka Ukuvinjwa umphumela yabo antihypertensive.

reception kanyekanye nabo "klopiksol" kungehlisa ukusebenza kwe-ejenti adrenergic, kuhlanganise "Levodopa".

Lapho kuhlangene izindlela abantu abazibheka "njengezijabulisayo piperazinyl" futhi "MCP" kwandisa ingozi izimpawu extrapyramidal.

izincomo ezithile

Izidakamizwa "klopiksol", intengo oboniswe ngezansi, ne ngokuqapha elibekelwe abantu nesifo senhliziyo, isifo sokusha kwesibindi kohlobo okungamahlalakhona, iziyaluyalu convulsive.

ukwelashwa isikhathi eside kufanele kube njalo ukuqashwa kokwelashwa ukuhlola isimo lesiguli.

Lapho ethola neuroleptics CSN angagcina ebulalayo. Izici eziyinhloko esesimweni esinjalo kukhona rigidity kwemisipha, ukuphazamiseka ukwazi, ukungasebenzi kwekhono NS autonomic, komzimba okukhulu.

Izindleko nokulungiselela libuyekeza ngakho

Inani kubhekwe izidakamizwa incike kundlela ukukhululwa. 2 amaphilisi mg e isamba yizicucu 50 ruble ngu-250, 25 mg (amayunithi 100) - ruble 1600, futhi 10 mg Tablets (izingcezu 50) - ruble mayelana 480.

Ngokuphathelene ikhambi uwoyela, amanani ayo ifinyelela ruble 2300.

Ngokuvamile, ukubuyekezwa yabathengi 'klopiksol "ukulungiselela ukushiya yalezo ziguli wasebenzisa izidakamizwa ngesimo umjovo. Iziguli ezinjalo abathi ukuthi izinga Ukusetshenziswa kwalesi thuluzi Kulula kakhulu ukusebenzisa. Lokhu kungenxa yokuthi imijovo kufanele kwenziwe akuvamile (njengoba kuqhathaniswa ngokuthatha amaphilisi).

Ngokusho kumpendulo yekhasimende, lesi sidakamizwa "klopiksol" kuyinto antipsychotic ngempumelelo kakhulu futhi fast-esebenza. Kodwa, ngeshwa, ngokuvamile kubangela engemihle.

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