ImpiloAmalungiselelo

"Ganaton": kumuphi umsebenzi, indlela yokwenza? Izibuyekezo "Ganaton"

Kuyini umuthi ezifana "Ganaton"? On yini eyenza leli thuluzi? Impendulo yale mibuzo itholakala kulesi sihloko. Uyofunda ngalokho umbono olwabiwa iziguli kule imithi, uma unazo Izimo, nendlela okufanele zithathwe ngendlela efanele.

Ifomu zomuthi, yayo emaphaketheni, ukubunjwa, incazelo

Ngayiphi ifomu ekhiqizwa izidakamizwa "Ganaton"? Imiyalelo, amazwana baphikisa ngokuthi ikhambi elinjalo angathengwa ngesimo amaphilisi, okuyinto asemhlophe, igobolondo (ifilimu), nxazonke wakhiwa, umbhalo «HC 803" ngakolunye uhlangothi kanti ingozi - ngakolunye.

Isithako asebenzayo we nomuthi kubhekwa hydrochloride itopride. Njengoba abamelwe asizayo buyisidakamizwa kuhlanganisa i-lactose, carmellose, corn isitashi, acid, silicic anhydrate, macrogol 6000, i-magnesium stearate, ama-titanium dioxide, hypromellose, futhi carnauba wax.

Ngo ukudayiswa izibhebhe ezinjalo ziza ibhamuza amaphakethe, nakho tihlelwe e amaphakethe amakhadibhodi.

Isimiso ezisebenza zomuthi

Siyini "Ganaton"? On yini eyenza lokhu izidakamizwa? Isetshenziselwa ukuthuthukisa motility emathunjini bese ithoni.

Njengoba isithako lokhu ejenti izenzo itopride hydrochloride. Le into izenzo ngokukhethekile endleleni engenhla wokugaya ukudla, futhi ngesivinini ukususwa ukudla esiswini. Kufanele kuqashelwe ukuthi le ingxenye yokubika iyakwazi ukunikeza umphumela antiemetic.

I izakhiwo zomuthi

Kuyini ephawulekayo yindlela ngokuthi "Ganaton"? On eliyenza, sizoqhubeka.

nomuthi Okubukwe kuyinto stimulator ukukhululwa acetylcholine. isithako Its main oyenza motility esiswini (ngamandla). Lokhu kungenxa umbango we Dopamine D2-yokwamukela kanye okusithiyayo umthamo ancike womsebenzi acetylcholinesterase.

hydrochloride Itopride oyenza acetylcholine kukhululwa, futhi kuvimbela nokucekelwa yayo.

izici Kinetic nomuthi

Lapho ukumuncwa onjalo izidakamizwa ngokuthi "Ganaton"? Yokusetshenziswa, ukubuyekezwa zithi ithathe isithako zomuthi ngokushesha kakhulu futhi cishe ngokuphelele kusukela esiswini. bioavailability wayo isihlobo cishe 60%. Lokhu kungenxa umzimba izidakamizwa, okuyinto eyenzeka ngo-pass lokuqala ngokusebenzisa isibindi. Ukudla ayinazo ukusebenza ngomhla ka-bioavailability ejenti.

Ngemva ukusetshenziswa (TEMLOMO) 50 mg itopride hydrochloride lokuhlushwa isiqongo kufinyelelwa kamuva 0.5-0.75 amahora imayelana 0,28 UG / ml. Okuphindaphindayo edonsa imithi ngesikhathi umthamo 50-200 mg kathathu ngosuku ngeviki pharmacokinetics komugqa. Kulokhu, ekuqongeleleni incane.

Ukuxhumana zemithi plasma amaprotheni cishe 96%. It is ngenkuthalo zisatshalaliswe ngazo zonke izicubu itholakala lokuhlala abaphakeme esikhathini isibindi, izinso, indlala adrenal, emathunjini amancane, futhi isisu. Imithi lingena kusivimbeli gazi ebuchosheni okuncane. Wabuye uyingqayizivele ubisi lukamama.

Excretion hydrochloride itopride nemikhiqizo yalo kwenzeka ne umchamo. excretion kwezinso we ketshezi esebenzayo ngemuva kokuthola umthamo owodwa zokwelapha imayelana 75%. Yokugcina isigamu-ukuphila kwalesi ejenti imayelana amahora ayisithupha.

Izidakamizwa "Ganaton": lokho kusiza?

Leli thuluzi is kabanzi ekwelapheni izinkinga gastro-emathunjini okuhlotshaniswa non-isilonda dyspepsia obusebenzayo (kuhlanganise kolwelwesi ezingamahlalakhona), kanye imisiwe motility esiswini.

Ngakho lapho ukusebenzisa izidakamizwa "Ganaton"? Isicelo sale izindlela siboniswa:

  • sokuzincisha;
  • ukuvuvukala;
  • isilungulela;
  • ukuhlanza;
  • uzizwa ekugcwaleni esiswini emva kokudla;
  • ubuhlungu noma ukungaphatheki esifundeni epigastric;
  • isicanucanu.

Enqabelo ukuze bathole imishanguzo engabasiza

Manje, niyazi, yini ephawulekayo yindlela ngokuthi "Ganaton". Kusukela lokho ephatha lesi ukulungiselela, siphinde ezitholakele. Kufanele kugcizelelwe ukuthi izidakamizwa kuncike is contraindicated ukuthola ku:

  • ukhulelwe;
  • ukopha emathunjini, isimiso mechanical noma perforation yokusetshenziswa pheshana emathunjini;
  • ngaphansi kweminyaka eyi-16;
  • ibele;
  • hypersensitivity kuya Itopride noma ezinye nezinsizasenzo imithi.

Qaphela ukulungiselela reception

Ithuluzi ebekiwe ngokuqapha abadala abantu ngenxa ukuncishiswa kaningi nezinso isibindi, kanye netifo concomitant noma ezinye ukwelashwa.

Ngenxa potentiation acetylcholine nomuthi kubhekwe ngokuqapha ukuncoma ukuthi iziguli ukuthuthukisa cholinergic side effects zingase zibe zimbi ngesikhathi isifo esikhulu.

Indlela "Ganaton"?

amaphilisi Kubhekwe okufanele zithathwe ngomlomo ngaphambi kokudla. Bahlanza phansi ngamanzi plain.

Umuthi akunamthelela ikhono lomuntu ukushayela izimoto, kanye izakhi eziyinkimbinkimbi. Uma usebenzisa "Ganaton" abantu abadala noma abantu kahle izinso umsebenzi futhi isibindi kubo kudinga kweso lwezokwelapha njalo.

Ngezinye izikhathi, udokotela afeze yokulungiswa umthamo Kunconywa. Uma ngephutha kugwinywe semali isidakamizwa edingekayo yokuqhuba ezifana izinyathelo ejwayelekile njengendlela yokwelapha isimo lingaze futhi lavage esiswini.

Ngayiphi umthamo isiguli kufanele adle imithi "Ganaton"? Isicelo (ukubuyekezwa imithi zichaziwe ngezansi) lokhu kusho ukuthi kudingeka kwenziwe ngemuva kokuxoxisana udokotela. Umthamo wansuku zonke zomuthi olucutshungulwayo abadala kuyinto 150 mg. Uma kudingeka, lemali ngenhla kungenzeka ashintshwe onekhono.

Njengomthetho, leli thuluzi Kunconywa ukuthatha kathathu ngosuku, iphilisi elilodwa ngaphambi kokudla (50 mg). Ubude yokwelashwa kunqunywa udokotela futhi kungase kube mayelana 5-8 amasonto.

isinyathelo uhlangothi

Wenzenjani ngokwemvelo kungabangela imithi "Ganaton"? Lokhu kusiza ikhambi sebuningini wokugaya ukudla izifo pheshana, kodwa kungase kumkhathaze miphumela elandelayo engathandeki:

  • Endocrine System: gynecomastia, amazinga prolactin anda.
  • uhlelo hemopoietic: thrombocytopenia, leukopenia.
  • komzimba: isikhumba ukulunywa, ububomvu kwesikhumba, anaphylaxis, ukuqubuka.
  • CNS: ikhanda, isiyezi, ukuzamazama.
  • ipheshana wokugaya ukudla: jaundice, uhudo, ngamathe yanda, ukuqunjelwa, ukucanuzela kwenhliziyo, ubuhlungu besisu.
  • Izinguquko nokuhlaziywa laboratory: anda amazinga bilirubin futhi ane-alikhali phosphatase, kanye umsebenzi ALT, AST kanye GGT.

izidakamizwa ekuhlanganyeleni

ekusebenzisaneni umzimba yalesi izidakamizwa akunakwenzeka. Lokhu kungenxa yokuthi itopride akheka isozymes akazange athonywe ka cytochrome P450, nangaphansi isenzo flavin monooxygenase.

Ingqikithi asebenzayo kubhekwa izidakamizwa kwandisa motility esiswini, okungase kuthinte ukumuncwa neminye imithi ngomlomo esetshenziswa kanyekanye. Isexwayiso Kufanele siqaphelisise lapho ukuthatha imithi nge Inkomba ongaphakeme zokwelapha. Kuyefana nasendleleni amalungiselelo ne enteric-camera okuqhubekayo-ukukhululwa ukwakhiwa kanye Isakhi esiyinhloko.

Lapho ngokuhlanganisa "Ganaton" nge "Diazepam", "warfarin", ticlopidine hydrochloride, diclofenac sodium, hydrochloride nicardipine futhi "nifedipine" izinguquko itopride ku sesibopho ukuthobisa plasma amaprotheni uyalandelwa.

Imishanguzo yama-isilonda ezifana "Ranitidine", "cimetidine", "cetraxate" futhi "teprenone" akuphazamisi kinetics we Itopride.

imithi Anticholinergic buthaka umphumela we ketshezi esebenzayo kokubuyekezwa izindlela.

Nutrition nokukhulelwa

Njengamanje, idatha enganele mayelana nokusetshenziswa Itopride hydrochloride ngesikhathi sokukhulelwa asipheli. Ukusetshenziswa leli thuluzi ngo-inqubo sokukhulelwa kungenzeka kuphela ukungabi kwamakhambi okwelapha, kanye olwanele ngezinzuzo umama, okuyinto mkhulu ingozi embungwini.

Kufanele kuphawulwe ukuthi ngesikhatsi ukwelashwa ngalo muthi kunobungozi amathuba okuba nemiphumela engemihle e usana. Kule ndaba, isidingo ukusebenzisa izidakamizwa esikhathini ukuncelisa ka lactation kufanele inqanyulwe.

izindlela ezifanayo futhi izindleko zomuthi

Ingabe uyasazi ukuthi kubiza malini phambi kwethu imithi? Uma ukwaziswa okunjalo okungekhona okwakho, sizokwenza yona. Intengo kwaleli thuluzi incike wekhasi, futhi inethiwekhi zosizo lokuqala imayelana 250 ruble amaphilisi 10.

Uma izidakamizwa alutholakalanga elinegama elifanayo, kungenzeka ukuba esikhundleni analogo. Phakathi leyo mithi ejenti ngalolu ketshezi asebenzayo afanayo, okungukuthi, ne Itopride. Njengoba ngokuvamile zisebenzisa "Itomed", "Itopride", "Itopru" futhi "Primer".

Izibuyekezo iziguli kanye nezifundiswa

Ingabe "Ganaton" nge Helicobacter pylori? Ochwepheshe ukubika ukuthi sikhuluma ngokuhoxiswa izindlela buyisidakamizwa esithuthukisa ithoni bese motility ipheshana wokugaya ukudla. Lena akuyona izidakamizwa elwa namagciwane ukuthi inganqoba igciwane oshiwo ngenhla. Nokho, kwezinye izimo namanje yaphathwa lesi sifo, kodwa ukwelashwa ngokuhlanganyela antibiotic namanye amanxusa anti-isilonda.

Cishe zonke iziguli abake kubhekwe ukuthi ngiphuza imithi, ukhulume kahle yaso ephezulu. Ngokusho kwabo, ngemva siwela inkambo yokwelapha izidakamizwa eqeda umuzwa nesicanucanu kabi esifundeni epigastric, kanye isisindo kanye nobuhlungu esiswini.

Ezinye iziguli isamukele lesi nomuthi njengoba kulungiselelwa nokuqedwa isilungulela episodic nokuhlanza.

Ngokuphathelene imibiko ukusabela ezingezinhle "Ganaton", ziyivelakancane. Njengomthetho, e seziguli ezithola lokhu ejenti kwezinye iziguli kukhulile amathe, ukozela noma isiyezi.

Uphenyo amacala ukweqisa izidakamizwa leli thuluzi engakaze fixed kuze kube manje. Intengo ekwakhiweni ezifana "Ganaton" ziqondakala abathengi njengoba isisebenzi esamukelekayo noma okusezingeni eliphezulu.

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