Impilo, Amalungiselelo
Umuthi 'Ketotifen': ukubuyekezwa kanye yokusetshenziswa
Izidakamizwa "Ketotifen" libhekisela eqenjini tsiklogeptatiofenonovyh izimali, okuyinto nethonya emelene histamine.
Lo mshini wezenzo zomuthi "Ketotifen"
Izibuyekezo odokotela abonisa ukuthi izidakamizwa kuvimbela ukukhululwa kwe histamine kusukela insika amaseli, zivimbela histamine receptor, kuthiye phosphodiesterase enzyme. Uma usebenzisa izidakamizwa kuwukwanda ezingeni ekamu e insika amaseli. Imithi ehilelekile nokucindezela platelet-isebenze isici imiphumela. Umuthi asisho ukukhiqiza ngempumuzo ukuhlaselwa isifuba somoya, kodwa evimbela ukubukeka kwabo kuphela, kunciphisa umfutho kanye nesikhathi, futhi kwezinye izimo, kuba zinyamalala ephelele. Umuthi kunomphumela omuhle isikhwehlela.
Ukwakheka kanye pharmacokinetics "Ketotifen" izidakamizwa
Izibuyekezo osokhemisi kanye yokusetshenziswa ibonisa e umuthi we-Isakhi esiyinhloko esebenzayo - fumarate ketotifen.
I nomuthi cishe ngokuphelele amuncwa wumzimba. I bioavailability we umuthi namaphesenti angu-50, kusho zokunqoba umgoqo gazi ebuchosheni. Umzimba kwenzeka esibindini, umuthi uboniswa ngendlela metabolites nezinso. Njengoba ingxenye enkulu yomsebenzi impahla egcina izinso esikhathini esiyizinsuku ezimbili.
Izinkomba lokwamukela "Ketotifen" ukulungiselela
Izibuyekezo nezeluleko odokotela elichaza imithi njengenhlangano usizo oluyilo ezinkantolo ekwelapheni ufuba atopic kanye dermatitis, hay fever, rhinitis iguliswa futhi conjunctivitis, futhi urticaria.
Umuthi ikhiqizwa ngesimo amaphilisi, 1 mg kanye isiraphu "Ketotifen".
Izingane ngaphezulu kweminyaka engu-mg ezintathu 1 kwezidakamizwa iqondiswa kunoma yiluphi uhlobo 2 izikhathi ngosuku. Abadala kufanele uthathe esilinganayo izidakamizwa ekuseni nakusihlwa. Uma kudingekile, umthamo kabili. Imithi ukusetshenziswa ngesikhathi sakusihlwa ngaphakathi. Isikhathi kwelashwa izinyanga 3. Ukuqedwa ukwelashwa wenziwa emavikini amabili.
Izimo futhi side effects ekuthatheni "Ketotifen" ukulungiselela
Nobufakazi ubonise ezifana izenzakalo ezimbi njengoba isiyezi, ukozela, kancane ukuphendula rates, umuzwa ukukhathala. Ngesikhathi ukusetshenziswa kwezidakamizwa siyenzeka ukupholisa, zingaphazamisa ukulala, kuphakama ukukhathazeka, uvalo ezinganeni. Ngaphezu kwalokho, iziguli ukuzwa nomlomo owomile, isifiso sokudla kakhulu bangase baqale ukuhlanza noma isicanucanu, ukuqunjelwa. ukusabela ezingezinhle ingase ihlanganise thrombocytopenia, komzimba, isisindo somzimba.
Izidakamizwa "Ketotifen", isiraphu kanye amaphilisi akunconywa lapho ekhulelwa noma ngesikhathi lactation. Kwenqatshelwe ngokuthatha izidakamizwa ezinganeni kuze iminyaka emithathu, kanye uma hypersensitivity kuya izingxenye.
Izidakamizwa "Ketotifen": imiyalelo ezikhethekile
Kuyinto engathandeki ukwenza yokukhansela abukhali zomuthi iziguli syndrome bronchospastic kanye isifuba somoya. Ukwelashwa kufanele simiswe kancane kancane, ukunciphisa umthamo ngaphakathi amabili kuya amane amasonto.
Iziguli nozwelo imiphumela sine kukhona, umuthi iqondiswa ngemithamo ongaphakeme. Imithi akuhloselwe ukwelapha bronchial somoya ukuhlaselwa. Ukuqokwa ahlangene ejenti hypoglycemic kufanele ukuqapha inani zegazi, okuyizinto igazi neuropathy.
Umuthi kuyalithinta ikhono izimoto netindlela ukuphathwa, ngakho kufanele uyeke lezi imisebenzi ngesikhatsi ukwelashwa.
Kusho icacisa imithelela elele amaphilisi, i-ethanol futhi antihistamine, futhi lihambisana imithi hypoglycemic kwandisa ingozi thrombocytopenia.
A imiphumela yempilo ezifanayo ube "Zaditen" izidakamizwa "Ketof", "STAF", "Positano".
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