Impilo, Amalungiselelo
"Terbinafine" (ukhilimu): yokusetshenziswa, analogs, ukubuyekezwa
Mycosis - lawa izifo ezibangwa isikhunta yisinanakazana. Sikwazi ukukhula esikhumbeni nesitsha nail, kanye izitho zangaphakathi.
Fungal ezingemnandi hhayi kuphela, kodwa futhi isifo esithathelwanayo. It is ngempela kalula ngocansi kusukela isilwane ukuze abantu futhi kusukela abantu esintu.
Namuhla kukhona imithi eminingi ehlukene ngempumelelo ukulwa nezifo fungal. Omunye ethandwa kakhulu kulezi Isidakamizwa "Terbinafine". Analogs ithuluzi, kanye ukukhululwa izinhlobo zawo, izakhiwo, kanye nezindlela ukusetshenziswa izokwethulwa ngezansi.
Ukwakheka, incazelo, emabhokisini Ukwakheka
Ngayiphi ifomu ukuthi likhiqizwa antifungal ejenti "Terbinafine"? Cream - lokhu akukona kuphela indlela imali. Kodwa ukuthi bemthanda iziguli.
1% ukhilimu "Terbinafine" nail ukhunta ukusetshenziswa sangaphandle ezimhlophe, ukuthungwa eyohlobo amandla isici iphunga.
Isithako asebenzayo we umuthi terbinafine hydrochloride. Futhi, njengoba excipients ngokudala wathi izindlela usebenzisa Gcoba i-Benzyl utshwala, cetyl palmitate, monostearate sorbitan, polysorbate 60, cetyl utshwala, isopropyl myristate, amanzi ahlanzekile kanye sodium hydroxide.
Ngo iphakheji sithengiswa iyi-ejenti antifungal, njengoba "Terbinafine"? Ukhilimu ithunyelwa aluminium amashubhu (30, 15 g), futhi ngo orange ingilazi izimbiza.
Ngaphezu kwalokho wathi isikhunta, wathi izidakamizwa ikhishwe ngendlela izifutho yokugcoba, amaphilisi, futhi isixazululo.
Izimpawu umenzeli yangaphandle
Uyini izidakamizwa "Terbinafine" (ukhilimu)? Manual ithi ejenti antifungal ukusetshenziswa ngezihloko ezihlukene. It has a ezibanzi spectrum umsebenzi antimycotic. Ngisho e lokuhlala encane izidakamizwa liveza umsebenzi fungicidal ngokumelene isikhunta, dermatophytes nesikhunta dimorphic. Ngokuphathelene imvubelo izimuncagazi, kuye ngokuthi hlobo zabo, bebheka bonke izidakamizwa angase abonise umsebenzi kokubili fungicidal futhi fungistatic.
mshini wezenzo
kanjani "Terbinafine"? Cream okushintsha ngqo ngendlela efanele usaqala synthesis begazi sterols ezenzeka isikhunta. Ekugcineni, lokhu kuholela ukuntula ergosterol kanye ukunqwabelana squalene kumaseli, okuyinto enomthelela enecala ngokufa kwabo.
Lo mshini wezenzo "Terbinafine" zingachazwa ngezinqubo okusithiyayo we epoxidase enzyme squalene esisogwini ulwelwesi cell we ukhunta.
Kufanele ukuthi izindlela wathi akuphazamisi P cytochrome 450, kanye umzimba hormone noma ezinye izidakamizwa.
izici kinetic
Ingabe izidakamizwa antifungal ugxile "Terbinafine"? Cream ukusetshenziswa ngezihloko ezihlukene is amuncwa 5%. Ngakho-ke, lokhu izidakamizwa uyakwazi kunethonya kuphela ukuchayeka azinakwa letindzala.
ubufakazi
Yini inhloso ezifana izidakamizwa ngokuthi "Terbinafine" ingasetshenziswa? Cream, intengo oboniswe ngezansi, ezinqunyiwe kulezi zimo ezilandelayo:
- zokuvikela kanye nokwelashwa kwezifo fungal kwesikhumba bushelelezi, fungal tesikhumba, ukhunta, kanye Jock ukuluma , kanye nezifo fungal ezinyawo, cuphuluza dermatophytes;
- ukwelapha ulele multi anemibala;
- ukwelapha imvubelo izifo zesikhumba, okuyinto zazibangelwa ukhunta Candida, kuhlanganise inabukeni amawala.
Izimo
Kwezinye izimo, awukwazi ukusebenzisa izidakamizwa "Terbinafine"? Cream, engesiyo inani lentengo eliphezulu kakhulu, kwenqatshelwe ukuyisebenzisa khona hypersensitivity kuya terbinafine noma iyiphi izithako asizayo ezakha izidakamizwa.
Qaphela nomuthi wathi ezinqunyiwe izifo semithambo occlusive zezinyawo, iminyaka okusithiyayo of umnkantsha hematopoiesis, ukwehluleka hepatic futhi kwezinso, izifo umzimba, ukusebenzisa uphuzo ngokweqile, izimila kanye nezingane ezineminyaka engaphansi 12 ubudala.
Njengoba lisetshenziswe ejenti antifungal "Terbinafine" (ukhilimu)?
Izibuyekezo ochwepheshe ukubika ukuthi lo mkhiqizo senzelwe kuphela lokusebenza langaphandle. It ingasetshenziswa kuphela ngoba iziguli omdala futhi intsha engu-12 ubudala.
Ngaphambi isicelo zomuthi okudingekayo ukuze ahlanze, bese ukuze ome izingxenye abathintekayo. Imithi esetshenziswa elilodwa noma amabili ngosuku. It sisetshenziswa ungqimba elincanyana ezindaweni ezithintekayo kwesikhumba kanye ezindaweni ezakhelene.
Kancane wagcoba ukhilimu, ukulishiya leli fomu, ngaphandle wokuwasha.
Ukuze izifo okuyinto ahambisana intertrigo, izindawo kwesicelo zomuthi ovunyelwe ukumboza gauze (ubusuku).
Uma kukhona umzimba olunzulu fungal izifo izidakamizwa Kunconywa ukuba isetshenziswe amashubhu 30 g
Isikhathi yokwelapha lokhu kusho incike uhlobo isifo fungal. Lapho umbandamu yomzimba, izinyawo nemilenze ukwelashwa wenziwa ngeviki, besebenzisa ukhilimu kanye ngosuku. Lapho candidiasis kwesikhumba futhi ezimise okwama-tile emibalabala izidakamizwa Kunconywa ukuba isetshenziswe amasonto amabili, lubricating kubo endaweni ethintekile kabili ngosuku.
Njengomthetho, ukwehla kwe izimpawu zokwelashwa izilonda fungal kuphawulwe ngezinsuku zokuqala yokwelapha. Ngekusetjentiswa okungajwayelekile imithi noma ukunqanyulwa kwanoma inqubo yokwelapha kukhona ingozi yokuphindela ukutheleleka.
ngemva Uma emva 2 amaviki Ukuqalwa okwelashwa, zimpawu zokuthuthuka bebelokhu akudingekile ukuba afeze ukuqinisekiswa uphethwe.
Isikali ezigulini esezikhulile akuyona ezahlukene kusukela ngenhla.
Sokuphuzisa spray "Terbinafine"
Futha "Terbinafine" isetshenziswa iziguli kaningi njengokuthanda ukhilimu. Ngokuvamile, leli fomu zomuthi kuboniswa for ekwelapheni izifo fungal izinzipho, isikhumba nezinwele.
Ngaphambi isicelo se-nomuthi isikhumba ngaphambili wageza obsushivayut. Ngaphezu kwalokho isetshenziswa endaweni ethintekile "Terbinafine". Futha wafutha ngendlela ukuthi ashutha kancane ingxenye enempilo kwesikhumba.
Ubude yokwelashwa nale ejenti kanye nokuvama ukusetshenziswa yayo incike kwasendaweni we ukhunta.
Kokudla izidakamizwa antifungal
Ayikho amacala ukweqisa izidakamizwa "terbinafine" ingakamiswa kubika. Uma ngephutha udle, singalindela ukuthuthukiswa ezifana side effects njengoba ikhanda, ubuhlungu epigastric, isicanucanu nesiyezi.
Ukuqeda lezi zimpawu sorbents ukunikeza isisulu, kanye nokwelapha bangisekela uma kudingeka.
izincomo Specific ukusetshenziswa ukhilimu
Ukuncishiswa izimpawu yesifo fungal kuphawulwe ngosuku lokuqala ukwelashwa. Isicelo okungajwayelekile ukhilimu noma ukunqanyulwa kwanoma yokwelapha, kunobungozi eliphezulu yokuphindela ukutheleleka.
Izidakamizwa "Terbinafine" senzelwe isicelo nezokusigcoba. Kufanele sizigweme ngamehlo nezinye nolwelwesi lwamafinyila, kungenjalo ngalesi siyingi kubangele ubuhlungu obunzima.
With ukuthuthukiswa komzimba ngokushesha kufanele uyeke ukusebenzisa ukhilimu.
Inani kanye analogue i-ejenti antifungal
Inani "Terbinafine" cream ruble mayelana 130-160 (15 g tube). Ezinye izinhlobo izidakamizwa ukukhululwa ungaba value ephakeme.
Umuthi ungayithola enye "Terbinafine"? Analogue kwaleli thuluzi etholakala ngazo zonke Pharmacy. Lezi zihlanganisa lokhu okulandelayo: "Atifin", "Bramizil", "Binafin" "Lamisil" "Lamitel", "Lamikan", "Mikonorm", "Onihon", "Mikoterbin", "Tebikur", "Terbiks", " Terbizil "," Fungoterbin ".
Umthengi Izibuyekezo mayelana izidakamizwa
Okwamanje, lesi sidakamizwa "Terbinafine" ngezindlela ezihlukahlukene ezahlukene ukukhiqiza enedumela elihle njengekhambi lokwelapha ephelele izilonda fungal kufinyelelwa ezimweni eziningi.
Ngokufanele ithuluzi, kunalokho ngokushesha aqede umuntu izinkinga edabukisayo.
Kepha nemibiko engemihle ke kungenzeka ashiye abantu awukagcwalisi uze uwaqede yokwelashwa noma imithi esetshenziswa ngendlela engavamile.
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