ImpiloAmalungiselelo

Codeine phosphate: yokusetshenziswa, analogs kanye nokubuyekeza

Codeine kungokwalabo umlaliso alkaloids chungechunge. It is kabanzi kwezokwelapha njengoba ikhambi for ukhwehlela. Libhekisela liphakathi oyibamba izidakamizwa okuyinto ngokuvamile sisetshenziswa ndawonye nezinye izinto, phakathi okuyizinto hydrate terpin. Ngempela ezithakazelisayo Kuyaphawuleka ukuthi ukusetshenziswa Codeine engaveza izimpawu izidakamizwa ukudakwa. imiphumela Kubhekiwe kanye analgesic. Kule ndaba, Codeine phosphate ingasetshenziswa ukuze kubulawe izinzwa, kodwa ngokuqinile by kadokotela.

Imininingwane emfushane

Umgomo we operation kuyafana Codeine ukuze morphine. Nokho, imiphumela yayo analgesic athé buthaka. Ndawonye nale phosphate Codeine (Latin lisho into njengoba codeinum) possesses kakhulu liphinyiselwe ikhono wehlise excitation ukukhwehlela isikhungo. Eqhubeka nalo mfanekiso ne-morphine, isibonelo, ukuthi kungcono kakhulu ukubuyeka ezicindezelayo umoya womuntu, hhayi kakhulu kuvimbela umsebenzi pheshana emathunjini. Naphezu kwakho konke lokhu, kaningi kukhona izimo lapho izidakamizwa kunomphumela Ugqozi emzimbeni, ekuvimbeleni ukozela.

Codeine phosphate: incazelo Izimo

Njengezinye imithi, Codeine inohlu umxhwele Izimo. Kufanele nakanjani babe nolwazi ngaphambi kokuba usebenzise izidakamizwa. Ukuze kwenziwe ngcono Umbono wakho, thina ukuhlukanisa nabo ohlwini ehlukile. Ngakho, i-izidakamizwa akufanele lisetshenziswe khona lezi zinto ezilandelayo:

  • hypersensitivity High;
  • arrhythmia;
  • ukuzibulala;
  • izinkinga emathunjini, wendlala indlala futhi urethra;
  • bekhulelwe noma lactation;
  • asebekhulile noma ubudala zezingane;
  • Kuye ukutholakala ketshezi izidakamizwa ebizwa phosphate Codeine;
  • isifo sohudo,
  • izinkinga umlutha wotshwala;
  • dispensiya anobuthi;
  • khona ukuhlaselwa isifuba somoya bronchial;
  • okulimala ebuchosheni, kanye izinso noma isibindi ukwehluleka.

Njengoba ubona, uhlu mikhulu. Ngokuvamile, ngaphambi ukusetshenziswa Codeine kufanele ngempela uxhumane nodokotela wakho. Ngeke libeke kadokotela ezidingekayo uma isimo somzimba wakho ikuvumela ukuba uthathe lo muthi.

Codeine phosphate: kanjani ukuthatha futhi kulokho ngemithamo?

Lapho usebenzisa i-Codeine ngezinhloso zokwelapha kufanele uqaphele ikakhulukazi uma kwenta tinhlaka umthamo efanele lomcebo, kanye nesikhathi wavuma. Ngakho, uma ubuhlungu acute kunconywa abadala ukuthatha 15-60 mg njalo emahoreni 3-6. Lapho sohudo kuyehla kube umthamo 30 mg kane ngosuku. Ekugcineni, lapho ukhwehlela nokuquleka kufanele baphuze 10-20 mg zomuthi izikhathi 4 ngosuku. Ephakeme umthamo zonke izinsuku we Codeine phosphate eye (ukubhala udokotela kadokotela) kuyinto mg 120.

Ezinganeni umthamo ukuhluka kancane. Ngokuvamile, isilinganiso iphelelwe 0.5 mg ngayinye 1 kg esisindo, uma kuziwa abacindezela izinhlungu ezihlukahlukene. Uma ukukhwehlela akufanele kuthathe ngaphezu 15 mg. Ekugcineni, sohudo njengoba umthamo kuyinto 0.5 mg ngayinye 1 kg esisindo. Ngokuphathelene ukuvama reception, kuba njengoba abadala, kufanele alingane izikhathi 4-5 ngosuku. By the way, izingane ezingaphansi kweminyaka ethola Codeine phosphate is hhayi Kunconywa engu-2.

imiphumela kwemithi

Njengoba kushiwo ngaphambili, Codeine kuyinto antitussive liphakathi esebenza. It kungokwalabo alkaloids phenanthrene yochungechunge. Ngaphezu kwalokho, liphinde iphathelene opioid yokwamukela agonists ezingaba kakhulu ukunciphisa excitability isikhungo ukukhwehlela, ngenxa okusithiyayo yayo eqondile. umsebenzi analgesic kungase kuchaze izidakamizwa ukusebenza opiate ezenza abonise excitation ezingxenyeni eziningi isimiso sezinzwa esiyinhloko. Plus, futhi sishintsha inombolo okuqonda ngokomzwelo ubuhlungu. Ngokuvamile, umphumela analgesic kuzibonakalisa emva kwemizuzu 10-45 emva umjovo, futhi nge isigamu sehora uma usebenzisa amaphilisi Codeine phosphate. Isikhathi senzo sithatha amahora ama-4.

side effects

Yiqiniso, Codeine phosphate has imiphumela engemihle, okuyinto wonke umuntu engaveza ngezindlela ezahlukene. Njengoba esimweni Izimo, sikunikeza uhlu imiphumela ngokuvamile azibonakali ngemva kokusebenzisa yalolu ketshezi:

  • Isimiso sezinzwa zinganqotshwa isenzo esinjalo: anda ukozela, ikhanda kanye nesiyezi (ezingavamile), kungenzeka ukusangana noma ukukhohlisa ezibukwayo, ukukhathazeka, amaphupho amabi ku amaphupho, ukucindezeleka (okuyinto ezingavamile), kanye nokuquleka. Lapho ukusetshenziswa amazinga okukhishwa ngokweqile bangezwa Isakhiwo sazamazama, Ukuwohloka ngefanelo nangokuvumelana futhi imisipha rigidity.
  • Ngo isimiso sokugaya ukudla bungene, miphumela elandelayo: isicanucanu nokuhlanza (akuvamile), ukuqunjelwa, amajaqamba esiswini, nomlomo owomile, kungenzeka anorexia futhi, ekugcineni, hepatotoxicity.
  • Cardio isimiso semithambo yegazi: arrhythmia, ukwehla okungazelelwe noma ukwanda wegazi.
  • uhlelo zokuphefumula: okusithiyayo eziqinile maphakathi kwemigudu yokuphefumula noma ukumelwa atelectasis.
  • Kukhona amathuba ukusabela elandelayo iguliswa: induna, ukuvuvukala kobuso nomphimbo, ukulunywa, bronchospasm, laryngospasm, futhi urticaria.
  • Ukuze ezinye imiphumela emibi evela ukusetshenziswa Codeine phosphate (ngesiLatini, ngenhlanhla umsindo codeinum) zihlanganisa ukujuluka ngokweqile, okuncane isimo sengeneme. Kanye ingozi sokuncika ngemigomo eside ukusetshenziswa (ikakhulukazi izinto eziningi ezinkulu).

Yiqiniso, ingozi olushiwo ngaphezulu side effects mncane impela. Yebo, futhi ngokuvamile ziyahlukahluka kusuka kokwenzayo esenzweni.

Izimpawu ze-ukweqisa izidakamizwa

zihlanganisa izenzakalo Izimpawu olandelayo ukweqisa izidakamizwa okungamahlalakhona: ukudideka engqondweni, isiyezi ezinzima, uvalo nolaka, Ukudlikizela, ubuthakathaka jikelele zomzimba futhi wegazi amathonsi. Ezimweni ezimbi kakhulu, kukhona awokuthi nokulahlekelwa ukwazi noma ikhoma kuqala. ukuphathwa Umlutha noma ukweqisa izidakamizwa isikhathi eside kakhulu futhi akulula. Ezimweni ubuthi kufanele iphume esiswini, ukubamba umoya wakhe futhi ukusekela umsebenzi inhliziyo. Kwezinye izimo, ngempela kunengqondo naloxone umjovo, okuyinto omelene ezithile analgesics opioid.

imiyalelo Special ngesikhatsi ukwelashwa

Lapho kukhona inqubo yokutakula ngemva Codeine ukweqisa izidakamizwa noma ukwelashwa ngenkinga yakhe, iziguli kufanele uyeke utshwala. Iqiniso liwukuthi ngesikhathi yokwelapha abantu kancane abathuntubezwe focus nesivinini lengqondo ukusabela. Utshwala kungenzeka senze isimo sishube namandla kuphela. Futhi ungaba nethonya elibi endleleni umuntu ekwenzeni imisebenzi engase ibe yingozi.

It kudingeka siyinake ngokukhethekile ngesikhathi sokukhulelwa kwabesifazane. Ngempela, ukusetshenziswa Codeine kungabangela ukubambezeleka Ukuqina sekuyenzeka, futhi ngezinye izikhathi ilethwe ngokushesha - prolongation. Ngokuvamile, amahlaya kanye ezimbi. Ekugcineni, njengoba kushiwo ngenhla, izingane ezincane, ngokuvamile, akufanele bathathe Codeine. Kulokhu, kukhona okungenzeka eside nesenzakalo ukusabela nakuba, njengoba izingane ziye zanda ukuzwela emiphumeleni analgesics opioid.

semthethweni

ERussia, kukhona manje bill, usebenza nezidakamizwa Codeine. Ngakho-ke, uyithenga ekhemisi ngaphandle kadokotela akukwazi. Muva nje, ukusetshenziswa Codeine isiko waqala wazise umphakathi, njengoba ukuthandwa izidakamizwa lukhula exponentially. Ngezindlela eziningi lokhu "sokunconywa" American hip-hop abaculi ngubani ngokuvamile ikhuthaza ukusetshenziswa Purple Drunk - isiphuzo ekhethekile equkethe ebulilini Codeine. isiraphu okunjalo has a luhlaza Pinkish-purple, futhi kungani lokho kwakuyisenzo igama obungajwayelekile. Ngemva ukuphuza ketshezi, uzohlangana umuzwa kwesasa omnene efana ecstasy opiates, okuyilokho, eqinisweni, libhekisela Codeine. Songs of rappers American ngokuvamile nombhalo, ekhomba ukusetshenziswa esihleliwe Purple Drunk. By the way, umdali bale nhlangano - Dj Intulo. Washona eneminyaka engu-29 kusukela ukweqisa izidakamizwa of Codeine.

Kufanele kuphawulwe ukuthi Codeine tholakala kweminye imithi, kuhlanganise zonke izinhlobo imfiva, protivomigrenoznye nabanye. Kule ndaba, imithi eminingi zivinjelwe ukudayiswa endaweni yeRussia. Futhi ukusatshalaliswa emthethweni futhi ukudayiswa kungaba uthole iminyaka engu-12 ebhadla ejele.

Ekuphetheni

Codeine has a ububanzi ezibanzi, njengoba nemiphumela yayo enkulu yomzimba womuntu yakhiwa enamandla kakhulu. Kungaba esikhathini kwetfulwe esifushane ngenhloso yokushintsha umqondo ogcwele we isimo somzimba umuntu. Uhlobo oluvame kakhulu Codeine (phosphate) - powder okuyinto kalula oncibilikayo emanzini. Ngenxa impahla yayo, liye kabanzi kusetshenziswa imithi. Nokho, njengoba kuye kwenzeke uma nge opiates, ketshezi seeped Khawuleza, uye emigwaqweni, okuyinto kunomthelela ongemuhle kubantu oqothulayo ke, imiphumela okungase ngisho ukubulala.

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