ImpiloAmalungiselelo

Antiplatelet ejenti "Clopidogrel": yokusetshenziswa

Kusho "clopidogrel" imfundo manual uchaza njengoba antiplatelet ejenti, esekelwe egcinwe ukwehla platelet wokuhlanganisa esibangelwa agonists ahlukahlukene. Ngaphezu kwalokho, lokhu izidakamizwa has a wawubona nomphumela vasodilatig. ukusetshenziswa isikhathi eside ka "clopidogrel" ukulungiselela (yokusetshenziswa igxile ukuthi ukunakekelwa okukhethekile) akuvumeli egazi ukuthi izinhlamvu ziqala ukwakheka amahlule, dala amahlukuzo lokubolekwa. Ngakho, ithuluzi kunciphisa ingozi yokufa uhlangothi nokumelwa yinhliziyo okwenzeka ezimweni lapho thrombus, kwakheka okuyinto engxenyeni emincane umfula, futhi kuvimbele ukugeleza kwegazi ligamanxa ukugeleza izakhi kanye nomoya-mpilo ezicutshini begazi.

Iyatholakala namuhla imithi "Clopidogrel" kuphela ngesimo round pink amaphilisi. Ukwakheka pellet ngamunye njengoba isakhi esiyinhloko sihlanganisa angu ayisikhombisa nanhlanu ka clopidogrel. Nezinsizasenzo kukhona izinto ezifana namafutha ocolisekileyo, isitashi pregelatinized, macrogol, lactose anhydrous, magnesium stearate futhi microcrystalline cellulose. Ukwakheka igobolondo yakhiwa polyethylene glycol 400 futhi 6000, hypromellose, ama-titanium dioxide, kanye ne-aluminium echibini.

Thatha iphilisi "Clopidogrel" yokusetshenziswa nguMkhandlu ukuze kuvinjelwe i-stroke, isilethikusebenza, thrombosis lemithambo neuropathy ezifana, okungazelelwe ukufa senhliziyo nezinye izenzakalo ischemic in iziguli isifo sokuqina kwemithambo yegazi. Ngaphezu kwalokho, lokhu izidakamizwa evame ukunikezwa abantu abanesifo lihambisana acetylsalicylic acid nokuvimbela okuthiwa "yezinkinga thrombotic" uma kwenzeka i syndrome acute yenhliziyo.

Sebenzisa kusho "Clopidogrel" yokusetshenziswa akuvunyelwe hhayi Kunconywa abantu ukusabela iguliswa clopidogrel noma ukungabekezelelani ngazinye iyiphi izingxenye asizayo eziqukethwe ngezithako zawo. Akufanele bathathe lezi amaphilisi iziguli acute ukopha (isb, izilonda peptic) noma ukwehluleka ezinzima isibindi. Uhlu Izimo esiqinile, ahluke kubo bonke ngenhla, zihlanganisa ukukhulelwa, ubudala ngaphansi iminyaka eyishumi nesishiyagalombili ubudala, futhi inkathi lactation. Endabeni lactase ukuntula noma ukungezwani ne-lactose efanayo ungathathi izibhebhe "clopidogrel". Ngokunakekela nangodokotela bababhekene nezifo zenhliziyo omkhulu linqume lokhu izidakamizwa iziguli kwathiwa unesifo "nokwehluleka ukusebenza kwezinso" noma "sibi yokwehluleka kwesibindi." Lapho zonke izinhlobo izimo zokucabanga okubangelwa isifo ukuthi kakhulu ingozi yezinye ukopha, kanye nokuthambekela kwabo futhi ungasebenzisi izidakamizwa "clopidogrel". Ekugcineni, it is hhayi Kunconywa ukuthatha leli khambi kanye nemithi "Warfarin" "Heparin", futhi okungezona steroidal izidakamizwa eqeda ukuvuvukala.

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