Impilo, Amalungiselelo
"Tolperisone": analogue, intengo, yokusetshenziswa
Izifo ezithinta uhlelo zemisipha kungenzeka spasm imisipha futhi anda ithoni. Iziguli ezingazweli ku-esesimweni esinjalo, kudingeka ukwelashwa okufanele esekelwe ukusetshenziswa imisipha relaxants. Odokotela bavame ukunquma "tolperisone." Analogue, intengo, yokusetshenziswa zomuthi ezocatshangelwa esihlokweni.
Nomuthi ne esebenzayo izidakamizwa tolperisone hydrochloride itholakala amaphilisi. I nomuthi eminye wanezela stearic acid kanye citric acid, kanye lactose futhi crospovidone.
imiphumela kwemithi
"Tolperisone" analogue imithi imisipha relaxants, abe isenzo emaphakathi. Mshini ithonya zomuthi emzimbeni bengayiqondi ngokugcwele.
"Tolperisone" inikeza izinzwa wendawo. Kuyaziwa ukuthi nomuthi ngenxa ketshezi asebenzayo ekhona Ukwakheka, aqede hypertonus imisipha, okubangela ubuhlungu iphele. Umuthi ngcono kwegazi neuropathy, antispasmodic futhi sifinyelele adrenoceptor ivimbela imiphumela, ke kuvimbela umsebenzi ingxenye caudal ka kumiswa reticular zobuchopho.
"Tolperisone" analogue, omqondofana ongaqeda gipertonus striated kwemisipha izinhlungu zibe futhi uqede ke kulezo zimo lapho izinkinga athuthukile ngenxa abhubhisa isifo semithambo noma entsefalopapii.
Ukuze linqume izidakamizwa "tolperisone"?
Odokotela linqume izidakamizwa "tolperisone" ebukhoneni okulandelayo:
- izifo ephelezelwa spasm kwemisipha, njengalapho i-stroke, ukuqina kwamathishu eqonda; phakathi lezi zifo - encephalomyelitis, myelopathy;
- isifo, okuyinto ukubonakaliswa dystonia kwemisipha; lezi zihlanganisa-cerebral palsy, nezinye izinhlobo encephalopathy;
- izinqubo ngenxa lapho abathintekayo uhlelo zemisipha, kukhona imakwe kwemisipha izinhlungu zibe; Lezi zihlanganisa isifo sokuqaqamba kwamalunga ezithinta amalunga omzimba esikhulu, futhi lumbago; izimpawu ezifana spondylarthritis, spondylitis.
Lapho lusetshenziswa ngezindlela "Tolperisone" analogs eziyinkimbinkimbi zisetshenziselwa ukwelapha acrocyanosis, ukuqina kwemithambo yegazi, isifo Raynaud sika, angiopathy.
Izimo ethola "tolperisone"
Umuthi akukashicilelwa ukuba abaneminyaka engaphansi kwengu-18 ubudala, iziguli ezinemishini myasthenia gravis, abesifazane azalele futhi ukufeza ibele, iziguli abangakwazi ukubekezelela i-lactose nezinye izingxenye ukulungiswa.
Manual iqukethe ezinye ukulinganiselwa. Esikhathini nokwelashwa kweziguli kahle isibindi umsebenzi nemithi izinso kusetshenziswe ngokuqapha okukhulu.
Ngezinye izikhathi "tolperisone" analogue esimisiwe ngesikhathi sokukhulelwa. Kodwa njengoba umphumela le mithi emzimbeni kwabesifazane abakhulelwe engakaze wafunda, ukusetshenziswa kwabo kungenzeka kuphela ezimweni lapho izinzuzo emzimbeni wentombi kuningi kunokomuntu ingozi embungwini. ukwelashwa imithi ngesikhathi senyanga yokuqala kudinga ukunakekelwa okukhethekile ukuze isimo umzimba wesiguli. Therapy "tolperisone" ibele kumisiwe okwesikhashana.
Ukusebenzisa "tolperisone": Isikali
I nomuthi senzelwe ukusetshenziswa yangaphakathi ngemva ukudliwa kokudla (ithebhulethi kuthathwe esiswini esingenalutho has a bioavailability ongaphakeme). Umthamo watusa for ukwelashwa kokuqala 50 mg izidakamizwa izikhathi 3 nsuku zonke. Ngokuhamba kwesikhathi, lenyuka 150 mg, kodwa hhayi kakhulu, kodwa kancane kancane. Imvamisa ukuphuza umuthi uhlala ingashintshiwe. Isikhathi sokuvivinya esigulini ngasinye kunqunywa ngamunye.
Umuthi ngalolu ketshezi esebenzayo ngaphansi kwegama tolperisone hydrochloride, analogs ekwelapheni iziguli ukuqeda iziphazamiso ezazingase nasemkhakheni isibindi noma izinso (Kusho ukukhanya) isetshenziswa ngokuqapha kakhulu futhi ezikhethwe ngokucophelela Ukweqiwa. Kukhona isidingo nokuqapha njalo sempilo yabo. iziyaluyalu Sinzima Uyi contraindication ukuba ukusetshenziswa "tolperisone."
side effects
Inani elikhulu Izibuyekezo kubonisa tolerability ezinhle yezingxenye eziphilayo ekhona yokwakheka izidakamizwa. Kutfutfukiswa ukusabela ezingezinhle ngemuva kokuthatha amaphilisi akuyona ovamile kakhulu. Kakhulu akuvamile, kukhona ubuthaka imisipha, ngezinye izikhathi kukhona ikhanda, futhi khona nomfutho wegazi ophezulu. iziphazamiso ezazingase zibe khona ku wamathumbu imikhuba, lapho kukhona isicanucanu nokuhlanza. Kusukela komzimba kungase kube khona angioedema, pruritus, urticaria emva kokudla "Tolperisone" ukulungiselela. Imiphumela engemihle futhi babe analogue.
ukweqisa izidakamizwa
Ayikho amacala ukweqisa izidakamizwa abikwe. Ngenxa ukuthatha umthamo sibe sikhulu kunesihlalo Kunconywa, angagcina hypotension, ukwephulwa okumelwe uphefumule futhi ukhulume inhliziyo umsebenzi. Ukuqeda ezinjalo ezidingekayo lavage esiswini kanye nokuqaliswa ukuphathwa (osekelayo, lingaze).
Izidakamizwa ukuxhumana "tolperisone"
Uma izidakamizwa isetshenziswa ne niflumic acid, ithuthukisa umphumela wawo. "Tolperisone" kwandisa umsebenzi "clonidine", izidakamizwa psychotropic, izidakamizwa ezinikeza izinzwa kanye muscle neuropathy relaxants.
"Tolperisone" analogue zingahlanganiswa nezinye izidakamizwa - kwezidakamizwa, kuhlanganise i-ethanol, sedatives, elele amaphilisi.
Lapho kuhlangene nezinye imisipha relaxants isenzo esifanayo okuyinto elihunyushwe ngokuthi "Tolperisone" amaphilisi, kudinga umthamo esincishisiwe agent.
Imithi kungathinta izidakamizwa umzimba CYP2D6 isoenzyme Ubamba lichaza, okwandisa ingqondo.
Analogs, izindleko zomuthi
Yini esikhundleni "tolperisone"? A ingumuthi omuhle futhi zithandwa kakhulu kuba "Mydocalm", uma kunesidingo ingasetshenziswa njengendlela esikhundleni ingxenye esebenzayo efanayo.
izidakamizwa Akwaziwa nezinye embodiments, njengokuthi "tizanidine" futhi "Sirdalud". Ngaphezu kwalezi mathuluzi, ungasebenzisa "Tizaludom", "Tizanilom", "Liorezalom" noma "Baklosanom". Kunenye esikhundleni - "tolperisone-OBL». Lo muthi ushibhile ukwedlula evame ukusetshenziswa "Mydocalm", okuyinto ingenye ethandwa kakhulu izidakamizwa analogue "tolperisone." Inani, analogue - ngesisekelo yokukhetha esikhundleni ezizuzisa kakhulu futhi ngempumelelo.
Iziguli babephathwa kwemisipha relaxant "tolperisone" ngokuyisisekelo aneliseke yi. ukusebenza kahle esiphezulu kuqashelwe ukususa spondylosis futhi spondylarthritis, ikhambi, uma kunesidingo, encephalomyelitis, eqonda sclerosis. Inani isilinganiso amaphilisi nge umthamo 50 mg RUB 140, ne umthamo 150 mg -. Ruble 190.
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