Kusho enesihloko esithi "Tranexamic acid" kuyinto izidakamizwa antifibrinolytic, isinyathelo eqeda ukuvuvukala kanye antiallergic, kanye liphinyiselwe umphumela hemostatic lapho bleedings okuyizinto ezihlobene ukwanda fibrinolysis. Emongweni umuthi lo okusithiyayo of plasminogen Activator futhi plasmin okusithiyayo kwetinhlavu peptides asebenzayo futhi kinins abahileleke ngokuqondile ukusabela ukuvuvukala kanye nomzimba. Ngaphezu kwalokho, ithuluzi ezifana "Tranexamic acid", kakhulu yinde isikhathi thrombin. Ngokuphathelene izici pharmacokinetics zomuthi anti-fibrinolytic ngemva kokungenisa ke amuncwa umzimba 30-50% of nokushintsha kokudla nokufakwa yayo sokuqala, amazinga aphakeme waphawula plasma lokuhlala eziyikhulu namashumi - imizuzu eziyikhulu namashumi ayisishiyagalombili futhi ngemva kokusebenzisa. umphumela Antifibrinolytic ezicutshini walondolozwa ukuze nanhlanu - amahora nesikhombisa, ne-plasma - amahora eziyisikhombisa noma eziyisishiyagalombili ngemva nokuphathwa izidakamizwa "Tranexamic acid". Intengo leli thuluzi ruble mayelana 1300, futhi ungakwazi ukuthenga it in cishe njalo ikhemisi.
izidakamizwa Antifibrinolytic ikhiqizwa ngesimo izibhebhe milligram amabili namashumi amahlanu noma anamakhulu mahlanu, njengoba isixazululo umjovo, kanye isixazululo senzelwe abaphathi ngomlomo. Konke okungenhla umthamo amafomu afaneleka kahle ukwelapha nokuvimbela ukopha, sokucasuka nokwanda fibrinolysis jikelele. Ngokwesibonelo, i-ejenti kaningi iqondiswa, ngemuva kwalokhu ozobizwa "Tranexamic acid" e izimila abulalayo we wendlala noma amanyikwe, wegazi, ukungenelela kuhlinzwa ezithweni kwesifuba, ne izifo zesibindi. ukususwa manual umzanyana kanye kwangemva kokubeletha ukopha zifakwe ohlwini izinkomba eya endaweni. Ngaphezu kwalokho, ukusetshenziswa kwezidakamizwa "Tranexamic acid" kumele haematuria, angioedema, dermatitis nomzimba, eczema, ezinobuthi futhi izidakamizwa amawala, isifuba. Ngaphezu kwalokho, lokhu izidakamizwa kuboniswa ngenxa pharyngitis asebenzayo, laryngitis, namathansela, stomatitis, acinene, lesizalo futhi ukopha esiswini, ukukhishwa izinyo in iziguli ukuthi nginesifo oluhambisana diathesis. Njengoba kahle ithuluzi ezifana "Tranexamic acid", nge nyanga zonke, ngaphandle ezinkulu.
Ngokuqondene lokusebenza oluthile nemithi sokuphuzisa, esimweni ngasinye bededelwa ngamunye, esekelwe elinikeziwe isimo emtholampilo. Nokho, njengoba umthetho, ngesikhathi uvunyelwe ukuthatha ku akukho kuka 1-1.5 amagremu. Kulokhu, ukusetshenziswa kaningi kuyizikhathi ezimbili kuya kwamane ngosuku, kanti isikhathi yokwelapha - kusukela ezinsukwini ezintathu kuya nanhlanu. umthamo owodwa kwezokuphatha emthanjeni kuyinto 10-15 mg / kg.
I Izimo eziyinhloko ukusetshenziswa kwaleli thuluzi kukhona izimo ezifana ukopha subarachnoid, thromboembolism, ukwehluleka kwezinso, kahle ukubonakala kombala, futhi deep vein thrombosis. Ngaphezu kwalokho, akufanele usebenzise lesi imithi uma hypersensitivity ngabanye noma ukukhulelwa. emibi ehambisana edonsa ejenti anti-fibrinolytic, ibonakaliswe njengeyenziwe isiyezi, ukozela, hypotension, tachycardia, ubuthakathaka, futhi ubuhlungu besifuba.