Ezempilo, Amalungiselelo
"Desal": imiyalelo yokusetshenziswa, incazelo, amafomu okukhululwa, ukubuyekezwa
Kufanele ngisebenzise kanjani uDezal? Imiyalo yokusetshenziswa, izinkomba zokusebenzisa leli thuluzi kuzoxoxwa kulokhu kulesi sihloko. Futhi, uzofunda ngamafomu lapho umuthi ungathengwa khona, ukuthi usebenza kanjani emzimbeni womuntu nokunye.
Amafomu okukhululwa, incazelo yokulungiswa, ukwakheka kwawo kanye nokupakishwa
Phakathi kweziguli, ethandwa kakhulu yiwona amaphilisi avela kuDelizal. Ehlanganiswe ngesikhumba sefilimu, iqukethe izinto ezisebenzayo, njenge-desloratadine. Ngaphezu kwalokho, ukulungiswa kufaka phakathi izakhi ezisizayo ezinjenge- magnesium stearate, i- microcrystalline cellulose, i-talc, isitshalo se-corn esinezimboni kanye ne-mannitol.
Amathebulethi okuthengisa emaphaketheni wekhadibhodi ngezinhlamvu eziyi-10 noma ezingu-30.
Ngaphandle kwendlela yokwelapha ekhonjiwe, olunye uhlobo lwezidakamizwa elithi "Desal" lwenziwa. Isixazululo (imfundo ekusetshenzisweni kwe-agent izoxoxwa ngezansi) ibizwa ngephutha ngokuthi isiraphu. Kuyinto ecacile, engenambala futhi engenayo izinhlayiya zangaphandle. I-Desloratadine nayo ingumuthi osebenzayo wale fomu. Ngokuqondene nezinsiza ezisizayo, zihlanganisa ukunambitheka "tutti-frutti", i-sorbitol, i-disodidium i-disodium, i-propylene glycol, i-sucralose, i-citric acid monohydrate, i-hypromellose ne-sodium citrate dihydrate.
Isixazululo sezingane "Desal" (isiraphu) siqhubeka sithengiswa emabhodleleni weglasi elimnyama (50, 100, 60, 150, 120 noma 300 ml). Kuhlanganisa nesipuni sokulinganisa (5 noma 2.5 ml) noma umphakeli we-syringe (5 ml).
Izici zezemvelo zalesi sidakamizwa
Iyini imithi "Dezal"? Imfundo yokusetshenziswa ithi le antihistamine iyinhlangano agent esebenza isikhathi eside. I-Blocker ye-histamine yangaphandle ye-H1 receptors. Into esebenzayo yalesi sidakamizwa iyinhloko ye-metabolite esebenzayo ye-loratadine. I-Desloratadine ivimbela ukusabela kokumangalisa, futhi ikhulula ama-cytokines nama-chemokines angenawo ama-inflammatory.
Ngenxa yokwakhiwa kwamakhemikhali, isidakamizwa esithi "Desal" sivimbela ukuthuthukiswa kokuphendula okweqile, kuvimbela ukugeleza kwazo, kunomphumela wokulwa nokuhlaselwa kwe-anti-sturitic, kuvimbela ukuthuthukiswa kwe-edema yamathambo, kunciphisa ukuguqulwa kwama-capillaries, kuvimbela ukuqhuma kwemisipha ebushelelezi.
Omunye akanakusiza ukusho ukuthi imithi ebuzwayo ayinayo umphumela omubi kwisistimu yezinzwa, ayinayo impikiswano yokudambisa, ayithinti ijubane lokuphendula kwengqondo futhi ayibangeli ubuthongo.
Isenzo sezinto eziyisisekelo siqala imizuzu engu-30 ngemuva kokungenisa futhi siqhubeka usuku lonke.
Pharmacokinetics yomuthi
Isidakamizwa esithi "Desal" sithatha isikhathi esingakanani? Ochwepheshe bathi emva kokuthatha imithi ngaphakathi kwe-desloratadine ixhumane ngokushesha ngokwanele ukusuka endleleni yokugaya. Kutholakala egazini ngesigamu sehora, kanti ukuhlushwa okuphezulu okufinyelelwe kufinyelelwa cishe emahoreni amathathu.
Ukuxhumana nama-protein kuwu-85-89%. Ukudla ngesikhathi esisodwa kwamanzi noma ukudla akuthinti ukusatshalaliswa kwe-desloratadine nganoma iyiphi indlela. Akungena ngaphakathi kwe-BBB.
Isigaba esibulalayo se-half-life amahora angu-27. Isidakamizwa siboniswa njengesakhi se-glucuronide kanye namazinyo kanye nomchamo.
Izinkomba zokusetshenziswa
Ubeka nini umuthi "uDezal"? Imiyalo yokusetshenziswa ikhombisa ukuthi le mithi isetshenziselwa ukunciphisa, kanye nokuqeda izimpawu ezilandelayo:
- I-Urticaria, kubandakanya ukuchithwa nokwehla;
- I-rhinitis ye-allergen, kuhlanganise nokukhipha, ukuminyanisa kwamanzi, i-rhinoorrhea, ukuvuza emakhaleni, ukushaywa kwelungu, ukuluma nokubomvu kwamehlo, ukulila.
Ukungahambisani nokusetshenziswa kwemithi
Lesi sidakamizwa asikwazi ukuphathwa uma:
- Ukuncelisa;
- Ebusheni (iziguli ezingaphansi kweminyaka engu-12);
- Ukukhulelwa;
- Ukuphefumula kunoma yiziphi izinto zomuthi.
Futhi kufanele kuqashelwe ukuthi ngokunakekelwa okukhethekile i-agent ekhonjiwe inqunyelwe ukwehluleka kwenkunzi (okubi).
Imithi "Ukufuna": imiyalelo yokusetshenziswa
Ngumiphi umthamo onquma ukuthi umuthi "uDezal"? Efomu elibhekiwe, umuthi onjalo uthathwa ngomlomo, kungakhathaliseki ukudla kokudla. Kwabancane, kanye nabantu abadala, imithi inqunyelwe ama-5 mg noma ithebhulethi eyodwa kanye ngosuku.
Ngokuqondene nesisombululo, ibuye iphindwe ngaphakathi, kungakhathaliseki ukudla ukudla. Izingane ezineminyaka engu-1-5 zinika 2.5 ml isiraphu kanye ngosuku. Izingane ezineminyaka engu-6-11 zishiwo 5 ml yesisombululo kanye ngosuku. Intsha kanye nabantu abadala bavunyelwe ukuthatha u-10 ml wezidakamizwa.
Overdose
Ngokusho kwemibiko yezobuchwepheshe, isidakamizwa esithathwe esilinganisweni esidlula umthamo onconywe ngezikhathi ezingu-9 asizange sibe nemiphumela emibi. Nokho, ezimweni ezingavamile, iziguli zaqala ukulala. Njengokwelashwa, ukugcoba esiswini kuyasetshenziswa. Futhi, isiguli singabelwa ukwamukelwa kwekhabhoni esebenzayo.
Ukuphendula okubi
Njengoba kuboniswe ukubuyekezwa kweziguli, ukuthatha le mithi kungabangela imiphumela emibi. Phakathi kwezinto eziqashelwa kakhulu yizinto ezilandelayo:
- Ama-Hallucinations;
- Usizi, ukulala, ukulala nokugula kwengqondo;
- Ubuhlungu besisu, i-dyspepsia, i-nausea, isifo sohudo nokuhlanza;
- I-Tachycardia ne-palpitation;
- Ukushisa kwesifo sofuba, ukwandisa umsebenzi we-bilirubin nokusebenza kwe-enzyme yesibindi;
- I-Myalgia;
- I-Anaphylaxis, itching, i- angioedema, i- hives ne-rashes.
Ukusebenzisana kwezidakamizwa
Kuze kube manje, ukusebenzisana okunempilo nezinye izidakamizwa akuzange kubonakale (kuhlanganise ne- "Erythromycin" ne "Ketoconazole").
Kumele kuqashelwe ukuthi imithi esebenzayo yalesi sidakamizwa ayikhulisi imiphumela ye-ethanol ohlelweni lwezinzwa.
Ukubamba nokukhulelwa
Inhloso yesidakamizwa esibuzwayo ngesikhathi sokukhulelwa ayinconywa, ngoba ayikho imininingwane yomtholampilo ekuphepha kokusetshenziswa kwayo kule nkathi.
I-Desloratadine ingena kalula ebisi lwebele. Kulokhu, ukusetshenziswa kwalo ngesikhathi sokulahlwa kuvunyelwe.
Imiyalo ekhethekile
Uma isiguli sinomsoco omkhulu we-renal, isidakamizwa esithi "Desal" kufanele siphathwe ngokuqapha okukhulu.
Isidakamizwa asinomthelela emandleni omuntu wokushayela. Kodwa-ke, kufanele kukhunjulwe ukuthi akuvamile ukuba ezinye iziguli zithole ukulala. Kulesi simo, kufanele kuthathwe ukunakekelwa ngokweqile uma ushayela futhi usebenza nemishini eyinkimbinkimbi neyingozi.
Ama-analogues kusho, intengo yomuthi
Isidakamizwa esiphikisayo sokuthi "uDezal" singathengwa kunoma iyiphi ikhemisi. Kumele kuqashelwe ukuthi inani lalo liphakeme kakhulu (ngokusho kweziguli eziningi). Amaphilisi angu-30 kuyodingeka ukhokhe cishe ama-ruble angu-360 eRussia. Cishe izindleko ezifanayo yilo muthi futhi ngesimo sesisombululo.
Uma isiguli sinomuthi ophikisanayo othi "Desal", khona-ke ungashintshwa yi-analog. Imikhiqizo yezokwelapha elandelayo ibonakala ngokubunjwa kanye nesenzo esifanayo: Desloratadine, Nalorius, Lordestine, Ezlor no-Eliseus.
Ngaphambi kokufaka esikhundleni se-agent enqunyiwe nge-analog kubalulekile ukubonisana nodokotela. Lokhu kungenxa yokuthi imithi enjalo ingaba neminye imiphumela emibi kanye nokuphikisana, kanye nemingcele nezindlela zokusebenzisa.
"Desal": impendulo yesiguli
Ngaphambi kokuthatha le remedy ye-allergies, sincoma ukuthi ufunde ngokucophelela imiyalelo enamathiselwe, kodwa futhi nempendulo yesiguli. Ngololu lwazi, ungafunda ukuthi ungathatha kanjani kahle izidakamizwa embuzweni nokuthi yiziphi izilinganiso.
Ukubuyekezwa mayelana nesidakamizwa "Ukufuna" (kusuka emithanjeni) kuningi kakhulu. Iziguli zithi ngemva kokuthola izidakamizwa eziningana, izimpawu ze-urticaria ziyanyamalala masinyane, isikhumba sibheke futhi sishabalale. Futhi lo muthi uphulukisa ngokuphelele i-rhinitis ye-allergen. Ngokushesha kususa ukuvinjelwa, ukushaywa emakhaleni kanye nezinye izimpawu zesifo.
Noma kunjalo, ngaphezu kokuhle, le mithi nayo inezibuyekezo ezingalungile. Ngokusho kwabo, akusizi ngalutho, futhi ngezinye izikhathi ayinayo impumelelo ekuphenduleni okwenziwe okweqile.
Ochwepheshe bathi lokhu kwenzeka kuphela ngokusebenzisa kabi imithi, kanye nokungabikho kokuzizwa komzimba ngokwayo. Ngakho-ke, ngaphambi kokusebenzisa le remedy, kufanele njalo uxoxe nodokotela bese uthola ukuhlonza okuqondile (okungukuthi, thola ukuthi unesifo sofuzo noma esinye isifo esizibonakalisa ngendlela efanayo). Ungaguli!
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