ImpiloAmalungiselelo

Kuyini phenobarbital? Izinkomba kanye analogs izidakamizwa

Manje ambalwa abantu bazi ukuthi phenobarbital, nakuba yalolu ketshezi itholakala izidakamizwa amaningi athandwayo. Abantu abaningi bathatha iminyaka "Corvalol" noma "Valocordin", ngingazi ukuthi izithako aqukethe le mithi. Ngemva muva phenobarbital isibaluli izidakamizwa eziyingozi futhi uvinjelwe kwamanye amazwe. A imali kwezindlu kusekelwe kuyo kancane kancane waqala kuzonyamalala emakethe. Manje lesi sidakamizwa "Phenobarbital" futhi analogue yayo zisetshenziselwa kuphela kadokotela. Phela, leli ingenye anticonvulsants esebenza kahle kakhulu sedatives.

Kuyini phenobarbital

Le nto kusukela iqembu barbiturates. Kunciphisa excitability izinzwa ebuchosheni futhi ukusabalala ezinzwa amaza e isithuthwane. Lapho umphumela wawo kwandisa ukugeleza calcium ion esitokisini, okuyinto enomthelela nokuncipha motor umsebenzi futhi ukunciphisa bushelelezi imisipha ithoni.

Okokuqala etholwe lokhu okubalulekile ekuqaleni kwekhulu lama-20 e-Germany. Sales phenobarbital sibonakala ngokuthi "Luminal". Kwakuwusuku ethandwa kakhulu ubuthongo usizo, ongakabi zaqhamuka ziphuma kule iqembu benzodiazepine izidakamizwa. Eminyakeni yamuva, amazwe amaningi ziye zathi ukukhiqizwa kwe phenobarbital. ERussia amalungiselelo okusekelwe kuso kukhona ukudayiswa, kodwa kuphela kadokotela kadokotela.

Manje ngokuyinhloko asetshenziswa "Phenobarbital" ekwelapheni isithuthwane. Futhi analogs yayo izindlela equkethe into ngesilinganiso esincane, ingasatshenziswa ngaphansi kwezimo ngaphansi ezinzima, ezifana ukuqwasha noma overexcitation.

umphumela iNarcotic yalolu ketshezi kuyinto ekhethekile: it akakubangeli kwesasa, ukozela nokunganaki kuphela. Ngaphezu kwalokho, yokwamukela phenobarbital kuholela kwencika enamandla kakhulu. Kodwa ukuthandwa okulahliwe kwakhe njengoba izidakamizwa kungenxa cheapness nokutholakala.

Amalungiselelo ngesisekelo phenobarbital

Umuthi elinegama elifanayo ejwayelene ikakhulukazi iziguli ezinokuphazamiseka convulsive noma izinkinga zokulala ezinzima. Kodwa ungakwazi ukuthenga izidakamizwa, ezibandakanya Phenobarbital. edume kunazo kukhona "Corvalol" futhi "Valokorin". Ziyakwazi ezishibhile futhi ethandwa kakhulu njengendlela okuyiluthayo futhi sine, ikakhulukazi isizukulwane amadala.

Ngaphansi adumile izidakamizwa ezifana:

  • "Lavokordin" ngaphandle phenobarbital, iqukethe valerian akhiphe, uwoyela peppermint futhi Uhobhane.
  • "Neo-Teofedrin" - kuyinto antispasmodic, elisetshenziswa somoya bronchial, iqukethe theophylline, i-caffeine, ephedrine, paracetamol.
  • "Paglyuferal" - izidakamizwa antiepileptic ngesisekelo phenobarbital.
  • "Pentalgin-N" - analgesic kwezidakamizwa.
  • "Piralgin" - lohlanganisiwe non-steroidal ejenti eqeda ukuvuvukala.
  • "Tetralgin" - isidambisa-zinhlungu futhi imithi antispasmodic.
  • "Andipal" - usetshenziswa njengesibonelo vasodilator e nomfutho wegazi ophezulu.

Izici yesenzo

amalungiselelo fenobaritala based Sekuyisikhathi eside kusetshenziswa imithi. Prescribers ngisho nezingane, ngoba izindawo eliyingqayizivele. Ngo pathologies ezithile kuphela ingasetshenziswa ukusiza isiguli. Isenzo phenobarbital sisebenza kuphela ku-imisipha bushelelezi futhi izinzwa ngaphandle kokuphazamisa yisimiso senhliziyo nemithambo yegazi. Lapho ethola izidakamizwa ezifana ngaphakathi imiphumela enjalo kuyagcinwa:

  • kancane encishisiwe ukushuba izinqubo umzimba;
  • kwehle motor umsebenzi;
  • It kunciphisa tonus kwemisipha abushelelezi pheshana emathunjini;
  • anda ngokukhishwa kobuthi egazini umsebenzi kwesibindi;
  • incipha lokuhlushwa bilirubin egazini.

Phenobarbital kabanzi imithi ngenxa yokuthi ukuthi anazo anticonvulsant, sine okuyiluthayo nomphumela spasmolytic. Isetshenziselwa ezimeni eziphuthumayo, njengoba ngesikhathi abaphathi ezingamahlalakhona ke zikwenza.

Phenobarbital: izinkomba ukusetshenziswa

Manje asetshenziswa izidakamizwa okusekelwe kuphela ezimweni ezimbi kakhulu. Basuke bengasaqondiswa engabelwe ukuqwasha abavamile. I izinkomba for ukusetshenziswa ithuluzi kukhona uthi ezifana:

  • isithuthwane kunoma yiluphi uhlobo;
  • isifuthefuthe ezahlukene;
  • chorea;
  • meningitis, ngqi;
  • utshwala ukuhoxiswa;
  • ukukhubazeka spastic;
  • ukuqwasha ezinzima;
  • kwempilo yengqondo;
  • perevobuzhdenie, ukukhathazeka.

Izimo

Naphezu kweqiniso lokuthi "ubufakazi Fenobarital 'kuyingozi kakhulu, akuzona zonke iziguli zithole ukwelashwa okunjalo. ekuphathweni contraindicated izidakamizwa esekelwe kule ndaba kulezi zimo ezilandelayo:

  • nge isibindi ezinzima nezinso;
  • myasthenia gravis;
  • anaemia;
  • sikashukela;
  • nokucindezeleka;
  • buthakathaka isimiso sokuzivikela ezifweni;
  • isifuba somoya bronchial;
  • ukuluthwa utshwala;
  • ukungabekezelelani ngabanye;
  • phakathi nokukhulelwa kanye lactation.

side effects

Amalungiselelo equkethe phenobarbital, ubheke izinto kwezidakamizwa. Ngaphezu kwalokho, zingabantu kakhulu umlutha, ngisho ukusetshenziswa short-term kungenzeka yabo side effects:

  • ubuthakathaka jikelele, isiyezi, asthenia;
  • ukudideka, inkulumo disorder;
  • ukusangana, amaphupho amabi;
  • nokucindezeleka;
  • iziyaluyalu ubuthongo;
  • kwehle acuity ezibukwayo;
  • nomlomo owomile, isicanucanu, ukuhlanza, kahle wamathumbu umsebenzi;
  • thrombocytopenia, ukuntuleka kwegazi emzimbeni;
  • palpitations, esingamahlalakhona senhliziyo ebuthaka;
  • ukwehlisa umfutho wegazi;
  • ukuqubuka, ukuvuvukala, dermatitis, pruritus;
  • iphika.

Yokusetshenziswa

"Phenobarbital" kanye amalungiselelo zifana ukubunjwa ekhiqizwa ngesimo izibhebhe 100 no-50 mg abadala futhi 5 mg izingane. Kuye inkomba kanye mode eyamukelayo udokotela utjho Isikali ezahlukene. Njengoba umuthi okuyiluthayo kudingeka baphuze 100 mg ngehora ngaphambi sokulala. Uma "Phenobarbital" iye enikezwa engayitholi njalo isiguli abanesifo sokuwa, kunconywa 50-100 mg kabili ngelanga. Njengoba amalungiselelo sine ngesisekelo izidakamizwa ezithathwe endaweni umthamo 50 mg 2-3 izikhathi ngosuku. Yehlisa umthamo watusa kubantu asebekhulile kanye neziguli kanye nemisebenzi isibindi nezinso kahle.

Izingane "Fenoarital" ukhombe izinkomba esiqinile. Umthamo kunqunywa udokotela ngekuya yobudala futhi ngezimo zesiguli. Linqume izidakamizwa for isigamu sehora ngaphambi kokudla izikhathi 2 ngosuku. Umthamo ngokuvamile ezifana: 6 izinyanga ukuba 5 mg, kuze ngonyaka - 10 mg, eminyakeni 1-2 - 20 mg, kuze iminyaka 4 - 30 mg, kuze iminyaka 7 - 40 mg, eminyakeni 7-10 - 50 mg, futhi engu-14 - 75 mg. Ngemva kulonyaka, umthamo we izidakamizwa Simila.

With ukusetshenziswa njalo kancane kancane kufanele umutsi. Lapho yokukhansela ngokuzumayo ngesisekelo phenobarbital izidakamizwa ngokuvamile ukuthuthukisa ukucindezeleka, ukuqwasha, ikhanda. Ukuthembela eba ngemva ukuvuma wemaviki lamabili njalo, it is hhayi Kunconywa ukuyisebenzisa njengendlela aid ubuthongo futhi sine izinsuku isikhathi eside kunaleso 10.

imiyalelo Special ukusetshenziswa

Abantu abaningi abazi ukuthi yini phenobarbital, kodwa buthule noma ukusebenzisa izidakamizwa kwezindlu kusekelwe kuyo. Ezinye zazo zidayiswa ngaphandle kadokotela, nabantu awazi ngisho kangakanani ezidakamizweni ezisebenzisayo. Ngakho-ke, kuyinto efiselekayo njalo ukufunda ukwakheka kanye imiyalelo ngaphambi isicelo izidakamizwa ngamunye. Uma usebenzisa phenobarbital ukulungiselela equkethe, kuyatuseka ukuba uhlole izici ezifana:

  • ketshezi aqoqana emzimbeni futhi kungakwenza umlutha;
  • ukwelashwa bayeka nalezi izidakamizwa kufanele kube kancane kancane, ngoba ngokuvamile kukhona "ukuhoxiswa";
  • lapho kuthathwe njalo akakwazi ukulawula imoto benze umsebenzi odinga ukunakekela nomsebenzi omuhle ukuphendula;
  • ngenkathi ethola nge izinto zokuvimbela inzalo temlomo, imithi elwa namagciwane, ama-ejenti antifungal incipha kahle kwabo;
  • Le into futhi kunciphisa digestibility glucocorticosteroids, anticoagulants, salicylates futhi estrogens;
  • ngenkathi ethola utshwala noma antidepressant angagcina okusithiyayo we isimiso sezinzwa esiyinhloko;
  • Le into kwandisa imithelela analgesics, imisipha relaxants futhi sedatives;
  • phenobarbital encishisiwe umphumela okuyiluthayo, lapho athathwa kanye Belladonna izidakamizwa atropine, thiamine, nicotinic acid izindlela psycho-ivuselela;
  • It akuvunyelwe nakancane ukuthatha le mithi sokukhulelwa, ikakhulukazi phakathi nezinyanga ezintathu zokuqala, njengoba lokhu kuholela ukuphazamiseka igazi ekunqandeni umntwana futhi ukubukeka ukopha;
  • ethola lactation phenobarbital kubangela okusithiyayo isimiso sezinzwa umntwana.

izidakamizwa analogue

Bambalwa abantu bazi ukuthi "Phenobarbital" amaphilisi. analogs ukuthi izimali zisetshenziswa kaningi. Sekuyisikhathi eside Isenzakalo esidume kunazo zonke kubo kube "Luminal". Kodwa muva nje, yena kuyaqabukela asetshenziswa. Kuyinto evamile ngaphezulu manje lezo zimali:

  • "Topirol".
  • "Zeptol".
  • "Barbital".
  • "Doxylamine."
  • "Sodium Etaminal."
  • "Orphir".
  • "Gabagamma".
  • "Depakine."
  • "Phenazepam".

Uphenyo pentobarbital

Odokotela abaningi abaphikisa ukuqokwa izidakamizwa ezinganeni ezingaphansi kweminyaka engu-6. Kodwa namanje wayevame ngisho kulonyaka ka phenobarbital. Izibuyekezo zale ndlela yokwelapha ayihlangani. Abaningi bathi inombolo enkulu yemiphumela emibi. Ngokwesibonelo, iziguli eziwohlokayo inkumbulo, ukucindezeleka eba. Abanye sokukhuluma kahle mayelana izidakamizwa, bekholelwa ukuthi into esemqoka - ukuze bagcine umthamo bese ulandela yonke izincomo udokotela. Iziguli enjalo ngesisekelo ezishibhile izidakamizwa phenobarbital (iphakethe kubiza ruble angu-20), futhi umphumela okuyiluthayo lokuhle kwabo. Kodwa amaphilisi enjalo okunikelwa kadokotela.

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