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Izidakamizwa Antihypertensive "Aritel": yokusetshenziswa

Medicine "Aritel" imfundo manual eyichaza ngokuthi i-ejenti hypotensive banezimfanelo liphinyiselwe izakhiwo antianginal futhi antiarrhythmic. Lesi sidakamizwa kuyinto abakhethayo beta 1 adrenoblokatorom futhi ayinaso abalulekile ulwelwesi eliletha ukuthula izakhiwo. Ukusetshenziswa kwezidakamizwa "Aritel" yokusetshenziswa okuyinto ngempela enikeziwe kule ikhithi, evumela indlela ephumelelayo ukunciphisa esivimba amanzi nomoya-mpilo ngokufunwa, ephansi plasma renin umsebenzi nokushaya kwenhliziyo, kokubili lapho esephumule futhi ngesikhathi umsebenzi. Ngokuqondene izici pharmacokinetic zomuthi, lokuhlushwa eyaqopha egazini waphawula ngemva kwamahora amabili kuya kwamathathu emva kokungenisa, nakuyo inxenye ukuphila amahora eyishumi kuya.

imithi Iyatholakala "Aritel", intengo njengamanje uyahluka ruble 80-150 ngesimo amaphilisi biconvex ophuzi. Isici esebenzayo ingaqukatha eyodwa pellet angu emihlanu noma eyishumi bisoprolol fumarate. Ekhuluma ewukuhlakanipha okwenziwe izingxenyana isinyathelo Kollidon CL, ludipress, magnesium stearate, MCC, Silica, corn isitashi, polyethylene glycol 4000, tropeolin "0", hypromellose, talc futhi titanium dioxide.

Sebenzisa ithebhulethi "Aritel" ochwepheshe batusa for the nokwelashwa kweziguli senhliziyo noma ifomu ezingamahlalakhona ephethwe yisifo senhliziyo. Lapho umfutho wegazi ophakeme futhi libonisa ukunikezwa kwemisebenzi kulowo ejenti anti-anginal. Futhi ngokuvamile esetshenziswa ne izidakamizwa kubhekwe ukuvimbela ukuhlaselwa angina esitebeleni.

Linqume antihypertensive "imiyalelo Aritel 'ukusetshenziswa is hhayi Kunconywa ukuba abantu ngaphansi iminyaka eyishumi nesishiyagalombili ubudala ukuhlupheka kusuka ifomu oyingozi noma ezingamahlalakhona ephethwe yisifo senhliziyo, edema yamaphaphu, bradycardia ezinzima, hypotension noma angina Prinzmetal. isifuba somoya bronchial, vimba sinoatrial, lactic umzimba, ukushaqeka cardiogenic kanye AV-block besigaba sesibili nesesithathu zifakwe ohlwini Izimo. Ngaphezu kwalokho, asikho isidingo ukusebenzisa lezi izibhebhe wokugoqa, ukwephula neuropathy kwegazi ohlelweni, pheochromocytoma, futhi hypersensitivity kuya beta-blocker. Sebenzisa izidakamizwa antiarrhythmic "imiyalelo Aritel 'ukusetshenziswa is hhayi Kunconywa kanyekanye nge Mao inhibitor futhi cardiomegaly. uqaphe kakhulu kumele kusetshenziswe lezi amaphilisi esingamahlalakhona kwezinso noma hepatic, i-hyperthyroidism, myasthenia gravis, AV-nokuvinjelwa ngowokuqala degree, isifo sikashukela, psoriasis nokucindezeleka. Ngaphansi kokuqondisa udokotela kokuthatha lesi iziguli antihypertensive abadala.

Ngokuphathelene imiphumela engemihle engase elihlobene ne amaphilisi "Aritel", esivame kakhulu kulo bayizinkulungwane ukutubeka komzimba, isiyezi, buthakathaka kwezicubu, ukukhathala, Alopecia, agranulocytosis, futhi ubuthulu. Ngaphezu kwalokho, ezinye iziguli akhononde cystitis, Ukudlikizela, conjunctivitis nokuqwasha.

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