Impilo, Amalungiselelo
"Formoterol": yokusetshenziswa, analogs, ifomu ukukhululwa, ukubuyekezwa
izinkinga Lung - lokhu nalesi asikona ukuntela. Abenzi kuphela ibakhathaze, isimo sibe sibi isimo sempilo, kodwa futhi kungase kubangele yezinkinga ezihlukahlukene. Ngokwesibonelo, isifuba somoya ingaholela ngisho nasekukholelweni ukuthi ukufa. Umuthi 'Formoterol "yokusetshenziswa ozokwethulwa ngezansi, nje ekwelapheni izifo zemigudu yokuphefumula. Nokho, phawula ukuthi isetshenziswa ukuba alwe ibanga ewumngcingo izifo.
Izici yesenzo izidakamizwa
Kusho receptor beta-adrenergic, okusho ikhono ukwandisa mafutha anciphisa isikhala esingaphakathi bronchial. Ngakho-ke kakhulu kubamba ukukhululwa kwe histamine futhi leykotrinov wamaphaphu izicubu. The main isithako kuyinto fumartata dihydrate.
Umuthi izenzo emizuzwini engu-5, bese umphumela walo omkhulu kufinyelelwa emva 2 h. Uma ebucayini permeability bronchial, umuthi kuhlale kusebenza amahora angu-10. Lokhu kwenza kube nokwenzeka ukuze kuxazululwe le ngezimo zesiguli isikhathi eside.
A ingxenye enkulu izimali ngemuva ephefumula zingene esiswini. Kukhona izingxenye futhi wafunda. Ingxenye-ukuphila umuthi cishe 13 amahora. izingxenye zalo zigcinwa futhi akheka esibindini. Ukuhoxiswa zomuthi umchamo. bioavailability Its 40%. A oketshezini olungenambala lwegazi ke sibopha 68%.
Kakhulu idokhumenti eziyisisekelo ngawo kufanele ufunde ngaphambi kokusebenzisa imali "Formoterol" - yokusetshenziswa. Ukukhululwa ifomu zomuthi akayedwa, zikhona eziningana: Amaphilisi nge powder powder alinganisiwe egabheni, i aerosol alinganisiwe. Kungakhathaliseki ukuthi iyiphi uthenge, umuthi isetshenziswa kuphela lapho ephefumula. kusho e ibhokisi ithengiswe.
Yiziphi izinkomba ukusetshenziswa khona
Uma usuvele abake basebenzisa "Formoterol" imfundo manual (imithi omqondofana ezocatshangelwa kamuva) kubonisa ibanga esincane kwezicelo. Ungakhetha lezi izinkomba ukusetshenziswa:
- Ukulapha nokuvikela ukuvaleka abukhali mafutha anciphisa isikhala esingaphakathi bronchial - spasm.
- Asthma. Kulokhu, lesi sidakamizwa akuyona ezinkulu, kodwa isetshenziswa kuphela ukusekela umzimba.
- ukucinana kwemithambo yomoya emaphashini.
- emphysema yamaphaphu.
- Umzimba ongezwani nezinto spasm bronchial. Iqiniso lokuthi izidakamizwa uyakwazi zivimbela ukukhululwa kwe histamine.
- ukuvuvukala Obstructive elingenhla ipheshana zokuphefumula, okuyinto kuhambisana ukwephulwa wabo emoyeni permeability.
Kwezinye izimo, umuthi akuvunyelwe?
Akuwona wonke umuntu angamukela "Formoterol". Yokusetshenziswa ukhuluma ngalezi Izimo:
- ukuzwela kakhulu okusezingeni eliphezulu ukuba izingxenye eziyinhloko noma ezengeziwe zomuthi ukuthi kungabangela ukuwohloka.
- ukukhiqizwa ngokweqile kwama-hormone i-ndlala yegilo - i-hyperthyroidism.
- ukwanda esimeme blood pressure.
- Bekhulelwe nangenkathi bencelisa. Iqiniso liwukuthi noma yimuphi ucwaningo kule ndawo kwenziwa. Lokho akwaziwa noma ingxenye enkulu excreted ngobisi. Ngakho-ke, uma umuthi usengaphansi okudingeka zithathwe, kungcono uyeke ukuncelisa ibele. Njengoba ukukhulelwa, it is konke ezinqunywa udokotela ukuba khona.
- Ukuphazamiseka isigqi inhliziyo: arrhythmia, tachycardia.
- Isifo senhliziyo. Ukuxhumana kwezidakamizwa ezithile kungase kuholele ezinkingeni esikhathini ventricles.
- Iminyaka engu-5. Eyezingane ezincane, wethule izidakamizwa sinzima kakhulu.
Imiphumela engemihle
"Formoterol" (yokusetshenziswa kukhona kuphakheji ngalinye) kungabangela abanye ukusabela ezingezinhle, nakuba amathuba abo liphansi njengoba ehlonipha imithetho izidakamizwa. Kungase kube imiphumela emibi:
- Kusukela isimiso sezinzwa: ubuhlungu futhi yelangabi e inhloko, ukundindizela, Ukudlikizela, ukuqwasha, uvalo ukukhathazeka anda.
- Cardio-semithambo uhlelo: anda inhliziyo noma izinga ukuphazamiseka ukushaya kwenhliziyo, i-angina, ukunciphisa okuqhubekayo noma ukukhula wegazi.
- On the ingxenye ipheshana wokugaya ukudla: isicanucanu nokuhlanza, ezomile nolwelwesi lwamafinyila emlonyeni, ubuhlungu besisu, Gastroenteritis (ukuvuvukala esiswini), dyspepsia (nobunzima ukugaya, okungase ephelezelwa ubuhlungu syndrome).
- Uhlelo zokuphefumula: izifo ezithathelwanayo ze- bronchi, sinusitis, pharyngitis, namathansela, isifuba somoya, izwi kahle.
- Okunye: ubuhlungu esifubeni, nokungezwani komzimba nezinto ezifana nokuqubuka, pruritus, ukushaqeka anaphylactic.
Izici isicelo izidakamizwa
Uma udinga ukuthatha "Formoterol" imfundo manual elikushoyo imithamo ezifana:
- Ngo somoya bronchial okudingeka ukwenze inhalations njalo ngemva kwamahora angu-12 ka-12 mg. Kuthatha umoya 1-2 kuphela. Ngakho, umzimba ukwesekwa wenziwa. Uma ukuhlasela kungenziwa senziwa ukuvivinya umzimba, kungcono ukuthatha izidakamizwa imizuzu engu-15 ngaphambi kokuqala umsebenzi ohlongozwayo, umthamo uyefana.
- Ukuze sisekele e obstructive isifo samaphaphu kufanele kwenziwe ephefumula kabili nsuku zonke 12 micrograms.
Qaphela ukuthi ungasebenzisa izidakamizwa emelelwa kungekho ngokuvamile ngaphezu kwesikhathi esisodwa njalo ngemva kwamahora angu-12. Okungukuthi, umthamo sangemihla kumele singeqi 24 mg. Ithuluzi yakhelwe kuphela lapho ephefumula. Uma udokotela uye ezinqunyiwe isidakamizwa "Formoterol" yokusetshenziswa (aerosol elisetshenziswe kaningi), ke ivimbela balithathe ngemithambo yegazi, intramuscularly noma ngaphakathi.
Uma kwenzeke ukweqisa izidakamizwa
Ufanele ukuphuza "Formoterol"? Yokusetshenziswa (kadokotela iyatholakala ekhawunteni kuphela imvume ekhethekile udokotela) kuyinto ebhokisini akuyona nje. It ngokucacile umthamo imithi. Kodwa uma ngenxa yezizathu ezithile wephule lezi ziqondiso, kungase kwenzeke yokweqisa. Ikalwe izibonakaliso ezinje: tachycardia, nomlomo owomile, ikhanda elibuhlungu, isicanucanu. Uma isikhathi akusho alungise lesi simo, kungenzeka, ngisho ukubulala.
Nge ukweqisa izidakamizwa of esiphuthumayo ukubiza i-ambulensi. Ukwelashwa kufanele kube lingaze. Kulokhu, ukusetshenziswa okuqhubekayo izidakamizwa imisiwe. Phakathi ukwelashwa kubalulekile ukulawula ukusebenza inhliziyo usebenzisa electrocardiography. Phakathi nenkathi emumva ukweqisa izidakamizwa isiguli kufanele kube ngaphansi ebhekiwe ongoti.
Izici nokuxhumana zomuthi nezinye izidakamizwa
Wena thatha "Formoterol"? Yokusetshenziswa (analogue abe Ukwakheka efanayo) iqukethe ulwazi mayelana nezici inhlanganisela yakhe nezinye izidakamizwa. Ngokwesibonelo, ngokuqapha kufanele kuqashelwe ngesikhathi kufakwa ngayo ejenti adrenergic.
ukunciphisa sokugembula potassium amazinga emzimbeni kungabangela inhlanganisela "formoterol" isisu, ama, kanye xanthine nemikhiqizo. Nokho, i-potassium akuyona isimo unomphela. Futhi yimuphi umthamo wemvula lemali zangaphandle kwalesi sakhi emzimbeni ayidingekile.
Zama ukuthatha leli imithi nge tricyclic antidepressant. Inhlanganisela ngayo beta blocker kuholela Ukuvinjwa mutual isenzo le mithi. Okungukuthi, bazuze kuzo ngeke, kodwa umonakalo lungase lube lukhulu ngokwengeziwe.
Co-ukuphatha amathuluzi ezifana "quinidine" "Dizopiramid" kungaba yingozi, ngoba wenza ukuthuthukiswa inhliziyo ventricular arrhythmias. Uma kukhona impendulo inhliziyo ukuthola usizo lwezempilo, bese-ke kufanele ngokushesha uyekwa.
Izixwayiso
"Formoterol" (ngesandla usuwazi) inezici ezithile isicelo:
- Ungasebenzisi izidakamizwa yokususa i kuhlasela somoya. Ukuze wenze lokhu, zikhona izindlela. Uma udinga "Formoterol" yokusetshenziswa (impendulo kwaba ikakhulukazi okuhle) lithi kuphela ibhekwa yokwelapha eziyisisekelo. Uma ngesikhatsi ukwelashwa unomuzwa wokuthi lesi simo sibhebhetheka, kufanele ngokushesha kudokotela.
- Musa ukuphuza lokhu kuze imithi esikhundleni corticosteroids. "Formoterol" ayinayo liphinyiselwe umsebenzi eqeda ukuvuvukala. Kulokhu, ukusetshenziswa corticosteroids kufanele baqhubeka ngaphandle ukunciphisa umthamo enqunywe udokotela wakho.
- Kakhulu ngokucophelela ukuba sikuqonde okuyiwa abesifazane ukuthi nginesifo lesizalo fibroids, kanye abantu abanesifo sikashukela.
- Akufanele kube ngokushesha ngemva reception ukushayela noma kumisebenzi ezidinga ukunakwa.
- Awukwazi ukusebenzisa izindlela ngesikhathi kwezidingo. Iqiniso ukuthi isithako main uyakwazi ukuba nomthelela ongemuhle lesizalo Kufinyeta.
Analogs nezici isitoreji
Ngokuvamile, iziguli uthanda nesifutho, equkethe umthamo owodwa-100. Isitolo kusho udinga kuphole futhi endaweni emnyama, kodwa akuyona efiselekayo iqhwa. elangeni akufanele iwe on ibhodlela. Ungayifaki imithi kude umthombo ukushisa.
Uma kungahambisani nalo izidakamizwa, ungase ufune bonana nodokotela wakho mayelana analogue. ungabahlukanisa phakathi kwabo kukhona: "Atimos", "Oxis", "Foradil", "Bronhoril", "Shadrin". Khumbula ukuthi owakho ukuthenga siphinde sithathe ezinye izidakamizwa bengayi.
Izibuyekezo futhi eshalofini yokuphila
Njengoba for izibuyekezo, abasebenzisi uthi nomphumela omuhle, okusheshayo nehlala njalo. Nokho, imithi samanje has a zibiza: ruble 1300-1600. Ingabe ukwazi ukukhokhela hhayi zonke iziguli. Nobufakazi ukubika ukuthi emva izidakamizwa yokusabela enobudlova spasmodic ze- bronchi akufanele kumakwe.
Impilo eshalofini izidakamizwa emelelwa kuyinto 2 iminyaka. Nokho, ngemva uvula nesifutho, kungaba ilahlwe kude ngemuva kwezinyanga 4. Vala noma yiziphi kungenzeka yokuthola umkhiqizo ezandleni zezingane. Ngemuva kwesicelo cap ibhodlela kufanele lusekelwe ngokuqinile ivaliwe.
Yilokho. Khumbula ukuthi zokuzelapha igcwele kuholele ekufeni. Hlala uphilile!
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