ImpiloAmalungiselelo

"Artrozan": analogue, imfundo kanye impendulo

Kanjani futhi kungani kufanele usebenzise izidakamizwa "Artrozan"? Imiyalelo, analogs nokubonakaliswa ngenjongo yaleli izidakamizwa uzobe kuchaziwe ngezansi. Siphinde ngikuxoxele kwindlela wathi nomuthi ikhiqizwa futhi lokunye, yini izingxenye afakiwe Ukwakheka kwabo, wathi kubo iziguli, njll

Ukuma, emabhokisini kanye nencazelo komkhiqizo, ukubunjwa yayo

Ngayiphi ifomu ke luyasetshenziswa izidakamizwa "Artrozan"? Analogue zalo kubhekwe umuthi ube izinhlobo ezihlukahlukene zokubusa ngesimiso ukukhiqizwa:

  • Tablets. Isithako asebenzayo of lo mumo kuphuma meloxicam. Futhi-ke yakhiwa izakhi asizayo ngesimo monohydrate lactose, colloidal Silicon dioxide, i-sodium citrate, povidone, amazambane isitashi kanye magnesium stearate. "Artrozan" amaphilisi (analogue Russian kanye angaphandle okusesihlokweni esithi) ungaba shades ezahlukene ophuzi. a Amalungiselelo anjalo ikhiqizwa ifomu ayisicaba isici futhi phakathi notch. It is zahlanganiswa ngo amashashaza, okuyinto ezibekwe ebhokisini amakhadibhodi.
  • A isixazululo esicutshini umjovo "Artrozan" (imijovo). Yokusetshenziswa (analogue yaleli fomu banikwa ngezansi) ihlinzeka ukuthi ingxenye izidakamizwa kufakwe njengoba eziyisisekelo izidakamizwa meloxicam. Ngaphezu kwalokho, ikhambi yakhiwa futhi izingxenye ezengeziwe ezifana sodium chloride, glycine, poloxamer, amanzi, Omunye izinyo lomhlathi sodium isixazululo hydroxide kanye glycofurol. Leli fomu zomuthi iyatholakala njengoba uketshezi esobala futhi ophuzi e ampules, phama amakhadibhodi amabhokisi.

Amafomu analogue nokwenza kwabo

I analogue ezilandelayo ingasetshenziswa lapho akunakwenzeka ukusebenzisa "ukulungiselela Artrozan ':

  • A isixazululo ujove esicutshini "Movalis". Isithako asebenzayo lokhu umuthi meloxicam (izingxenye asizayo: meglumine, poloxamer, glikofurfurol, glycine, i-sodium chloride, i-sodium hydroxide, amanzi d / s).
  • Ploskotsilindricheskoy ithebhulethi ifomu "Meloxicam". Isithako asebenzayo we umuthi meloxicam futhi (excipients: microcrystalline cellulose, i-lactose, povidone, sodium citrate dihydrate, sodium carboxymethyl isitashi, colloidal Silicon dioxide, i-calcium stearate).
  • Amaphilisi kanye umjovo "Melbek". Isici esebenzayo lokhu umuthi meloxicam (izithako ezincane: povidone, lactose anhydrous, magnesium stearate, microcrystalline cellulose, sodium citrate, crospovidone, colloidal Silica anhydrous).

Lo mshini wezenzo zomuthi "Artrozan" futhi analogue yayo. Pharmacokinetics

izidakamizwa "Artrozan" Indlela Isebenza? Analogs ngokwayo nomuthi eliqukethe kwakwakhe esebenzayo ezifana meloxicam, amelela oxicam nemikhiqizo. Bona kunethonya imiphumela eqeda ukuvuvukala by ekuvimbeni enzyme tsikooksigenazu-2 kanye zamagama prostaglantinov okuyinto abahileleke ngokuqondile umjikelezo we arachidonic acid.

Ngemuva kokufaka isicelo umsebenzi izidakamizwa ka balamuli ukuvuvukala, kanye permeability izindonga semithambo wehlise kakhulu. Ngakho kukhona ukuphendula kancane nge free radicals.

Umthelela analgesic imithi ngenxa ukwehla womsebenzi kanye nokuxhumana kwalapho prostaglantinov.

Iziphi izici ine izidakamizwa pharmacokinetic "Artrozan"? Analogs wathi izidakamizwa uqobo ukufinyelela lokuhlushwa esiphezulu egazini zingakapheli izinsuku 3-5. Ukuthaka imithi uxhumano nomsebenzisi kahle amaprotheni (cishe 99%). umzimba wabo senzeka isibindi, kuphumele 4 metabolite. Ngesikhathi esifanayo abazi ukudlala likhona iqhaza izinqubo pharmacodynamic.

Izidakamizwa excreted ku umchamo kanye endleni.

Izici esiyingqayizivele

  • Izidakamizwa "Movalis" has a imakwe umphumela anti-inflammatory kunoma iyiphi ukuvuvukala izingxenye ahlangene emzimbeni.
  • "Meloxicam" imithi. isinyathelo eqeda ukuvuvukala yaleli izidakamizwa Lihlobene nokubhekana ubuso okwehlisa ka umsebenzi enzymatic of Cox-2.
  • "Melbek" imithi kanye nezinye analogs libhekisela eqenjini NSAID.

Izinkomba Zokusetshenziswa "Artrozan" izidakamizwa futhi analogue yayo

Analogue izidakamizwa "Artrozan" futhi izidakamizwa nokubika uqobo aqoke izinkomba efanayo. Zonke izidakamizwa ngaphezu zenzelwe aphathe ezihlukahlukene ukuvuvukala emalungeni ephelezelwa ubuhlungu syndrome:

  • osteochondrosis;
  • e-osteoarthritis;
  • rheumatoid arthritis;
  • e myositis;
  • e ankylosing spondylitis;
  • radiculitis.

Izimo ukusetshenziswa kwezidakamizwa kanye analogue yayo

Kungaphansi kwaziphi hhayi izimo ungasebenzisa izidakamizwa "Artrozan" analogue lokhu izidakamizwa? Ngokusho imiyalelo, ngokucabangela nemithi ( "Artrozana", "Movalis", "Meloxicam", "MELBEK") ube Izimo ezilandelayo:

  • isilonda duodenal nasesiswini;
  • njengemithi yokungezwani komzimba nokuthile izidakamizwa ;
  • luvelo izidakamizwa izinto;
  • ukungabekezelelani emaqenjini NSAID;
  • ukopha pheshana emathunjini;
  • somoya;
  • yobudala engaphansi kwengu-15;
  • polyp e ngalo ingaphakathi acinene futhi ekhaleni;
  • kwezinso ezinzima, inhliziyo noma ukungakhuli hepatic;
  • hyperkalemia;
  • hemophilia;
  • lactation, nokukhulelwa.

kufanele Ngithatha kanjani imithi "Movalis", "Meloxicam", "Melbek" futhi "Artrozan"?

Analogue "Movalis", kanye nezidakamizwa "Meloxicam" futhi "Melbek" abelwa ku imithamo efanayo "Artrozan".

Amalungiselelo ngesimo amaphilisi iqondiswa kanye ngosuku ngezikhathi zokudla, kufanele uphuze amanzi plain. I umthamo wansuku zonke lezi izidakamizwa 7.5-15 mg (kuye ngokuthi isifo nobuhlungu umfutho).

Uma imithi ngeke kuthathwe ngomlomo ke odokotela linqume ujove esicutshini. Kulokhu, umthamo wansuku zonke futhi kufana 7.5-15 mg. Kulokhu, ukwelashwa ithoma nge umthamo encane bese lingezelelwe kuze nomphumela ofiselekayo. Kunconywa ukuthi aseqeli umthamo, kusukela kuleli cala, kungase kwandise amathuba okuthola i-ukusabela ezingezinhle.

Overdosing izidakamizwa

Lapho usebenzisa i-ebulilini izidakamizwa "Artrozan", "Movalis", "Meloxicam" futhi "Melbek" Izimpawu ezilandelayo kungenzeka isiguli:

  • ukuqunjelwa;
  • ubuhlungu epigastric (ukopha kungenzeka esiswini);
  • ukuhlanza nesicanucanu;
  • ukungakhuli ukwazi;
  • ukuboshwa zokuphefumula;
  • asystole;
  • iziyaluyalu kwesibindi nezinso.

Ukuqeda izici ezifana abathintekayo esiswini wageza chelators ukwabela.

Side Effects "Artrozana" futhi analogue yayo

Uma uthola izidakamizwa "Artrozan", "Movalis", "Meloxicam" futhi "Melbek" kaningi kukhona nalawo mathonya ezingathandeki, njengobuwula:

  • ukudla ukuqunjelwa, ukubhodla, izilonda esiswini, ukopha esiswini;
  • kwesibindi, enzyme isibindi kuphakame, ukwehluleka oyingozi kwezinso;
  • bronchospasm, angioedema, edema neuropathy;
  • tachycardia, anaphylaxis;
  • leukopenia, thrombocytopenia, ukuntuleka kwegazi emzimbeni;
  • ikhanda, ukudideka, ukozela, isiyezi, angaboni kahle;
  • esophagitis, iguliswa isikhumba ukusabela, photosensitivity, pruritus;
  • stomatitis, conjunctivitis futhi urticaria.

izidakamizwa ekuhlanganyeleni

amalungiselelo Kuhlanganiswe "Artrozan", "Movalis", "Meloxicam" futhi "Melbek" nezinye imithi kufanele niqaphele kakhulu. Ukuze uthole ukuthi esibekela amathuluzi ivumelekile nokwelashwa arthritis ikuphi, kufanele ngaso sonke isikhathi xhumana nodokotela bese ulandela imiyalelo afakiwe. By the way, ku izidakamizwa zokugcina ezibalwe izici ezilandelayo:

  • kuhlangene ingcindezi ukunciphisa kusho ukusebenza kahle kwabo kuyehla;
  • ngokuhlanganyela "Tsiklosprorinom" futhi isisu kwandisa ingozi nokwehluleka ukusebenza kwezinso;
  • lihambisana fibrinolytic, vitamin K abamelene, heparin futhi serotonin reuptake inhibitor e isiguli bangezwa ukopha.

Kufanele futhi kuthiwe imithi "Artrozan", "Movalis", "Meloxicam" futhi "Melbek" ngokucophelela okukhulu okuhlangana ngayo lithium amalungiselelo, amadivayisi intrauterine, nezinye ama-NSAID, "Kolestiramin" futhi "methotrexate".

izincomo Specific ukuthola Analogue

Ukusetshenziswa kwezidakamizwa ezingekho steroidal ekwelapheni amalunga omzimba kungase kufihle izifo ezingathi sína kwababhemayo ezithathelwanayo ezenzeka emzimbeni wesiguli.

A ukusetshenziswa eside izidakamizwa (amasonto engaphezu kwemibili) kudingekile ukwenza ukulawula isibindi kanye nezinso.

Uma umuntu nezici ezithile ukuze ukubonakala isilonda we duodenum noma esiswini, bese usebenzisa imithi "Artrozan", "Movalis", "Meloxicam" futhi "Melbek" kufanele kube ngokuqapha. Kulokhu-ke kungcono ukusebenzisa isixazululo kwezokuphatha esicutshini.

Uma uneminye imiphumela okuhlotshaniswa izinga esincishisiwe lengqondo ukusabela, kufanele ziyeke ukusebenza nge izakhi eziyinkimbinkimbi, futhi noma kunjalo hhayi ukushayela izimoto.

I Analogue izidakamizwa

"Artrozan" e ampoules kanye amaphilisi has analogue abaningi wemithi emakethe yesimanje (Russian kanye angaphandle). kumakhophi Main abalwe ngenhla. Kukhona imithi efanayo kungabandakanya:

  • "Matar"
  • "Elithi bi-Xico"
  • "Medsikam"
  • "Movasin"
  • "Lem"
  • "M-Kam"
  • "Mirloks"
  • "Mesipol"
  • "Amelotex"
  • "Melox"
  • "Melox"
  • "Moviks"
  • "Meloflam" nabanye.

Iningi eseduze Analogue "Artrozan" izidakamizwa umuthi "Movalis". Libuye libe NSAID. Leli thuluzi isebenza nemikhiqizo enolovoy acid. It has eqeda ukuvuvukala, antipyretic nomphumela analgesic.

Futhi, ngokuvamile kakhulu lesi sidakamizwa "Artrozan" esikhundleni "meloxicam" noma "MELBEK". Lena izidakamizwa ezingekho steroidal anti-inflammatory ukuthi babe analgesic, antipyretic nemiphumela ethile eqeda ukuvuvukala.

Konke analogs ngenhla zenzelwe ukuze banciphise ubuhlungu, okuyinto kubonakala izifo ezihlukahlukene emalungeni. Phakathi kwabo kukhona ngempumelelo ikakhulukazi kunzima, ngoba zonke ukubhekana ngokugcwele umsebenzi.

Kufanele kuqapheleke futhi ukuthi lezi izindlela babe efanayo emibi, kanye contraindications (bheka ngenhla).

Nobufakazi ngezidakamizwa

Abantu abaningi ushiye okubuyayo mayelana Atrozan izidakamizwa ' "," Movalis "," Meloxicam "futhi" Melbek ". Ngokusho kwabo, lezi imithi ayatholakala, kodwa kuphumelela kakhulu. Iziguli eziningi ku esikhathini esifishane ukusiza balahle ubuhlungu syndromes, okuyinto avele izifo ezihlukahlukene emalungeni.

Kufanele kuphawulwe ukuthi ekwakhiweni ithebhulethi le mithi nomphumela ofanayo njengoba ukuthi umjovo.

Kulaba minuses izidakamizwa "Atrozan" futhi okungenhla analogue kuyinto ukusabela latsite lavamile enqabayo kuphawulwe ngesimo esiswini izinhlungu, ubuhlungu bekhanda nesiyezi.

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