Impilo, Amalungiselelo
Analog "Memantine": incazelo, yokusetshenziswa futhi impendulo
"Memantine" - ingenye izidakamizwa, okuyinto ngempumelelo ezihlukahlukene komqondo kanye Alzheimer. Lesi sidakamizwa, okuyinto adamantyl esuselwe, iyatholakala njengoba amaphilisi kanye amathonsi ngomlomo. Umuthi elingathi sína, kungadala nemiphumela engemihle. Ngakho-ke, izihlobo eziningi zeziguli ukubuza udokotela ukukhetha Analogue "Memantine" ngomphumela akuyona zingaphansi kwakhe, kodwa ivikeleke nakakhulu.
izici umkhiqizo
Lo muthi ikakhulukazi ngokuthi "Akatinol Memantine" ezaziwayo. The main izidakamizwa esebenzayo ke - hydrochloride memantine. It has a nethonya elihle umzimba ubuchopho izicubu, ephumula imisipha futhi ethuthukisa ukusebenza kwengqondo. Ngenxa nokusebenzisa kwayo inkumbulo ethuthukisiwe, bandisa inkonzo ngokomzimba, ikhono lokufunda. Ahamba kahle amalungiselelo kokuba zithako uphakathi kwabantu abangenalo leli kwemisipha relaxants ziye benganhlanhlathi ukudlula emsipheni amaza kagesi sibe kwemisipha izicubu futhi uvimbele calcium iziteshi.
Yikuphi isinyathelo has izidakamizwa
Naphezu inani elikhulu contraindications side effects, kanye iqiniso lokuthi izidakamizwa okuthengiswa kuphela kadokotela, umuthi kuvamile impela, "Memantine". Inani, ukubuyekezwa, analogs futhi ikakhulukazi izenzo zakhe zaziwa kulabo izihlobo abaphethwe komqondo noma Alzheimer. Nokho, lokhu izidakamizwa Ungase futhi ube omunye umphumela:
- kunciphisa imithelela hypoxia palsy, oxygenates amaseli;
- ngcono cerebral ukugeleza kwegazi, kunciphisa vasospasms;
- It Unazo izakhiwo neuroprotective, ukuvikela izinzwa ekulimaleni;
- Kuvuselela isimiso sezinzwa ngu toning umzimba kanye nekufaka ligalelo ukusebenza umsebenzi kwengqondo;
- Ithuthukisa inkumbulo, ikhono ukugxilisa ingqondo;
- Kuyasiza ukuba babhekane nokucindezeleka, kujwayeleke kwemizwa;
- aqede kwemisipha izinhlungu zibe kubangelwa ukulimala izinzwa ingqondo.
Izinkomba ukusetshenziswa zomuthi
Noma yimuphi analog "Memantine" njengoba kusho ngokwayo, liphumelele obuhlukahlukene degree of ukuphazamiseka kwengqondo. Lokhu ungaboniswa ukushintshashintsha kwemizwelo, amehlo inkumbulo encishisiwe okuhlushwa, Ukuwohloka amakhono bokusungula. Ngokuvamile lokhu isimo lihlotshaniswa ukukhiqizwa enganele Dopamine. Ngasiphi yobudala ingavela izifo ngoba kuyo okudingekile ukusebenzisa "Memantine". Analogue, okuyinto Izibuyekezo bathi kahle zabo eziphakeme, iqondiswa kulezi zimo ezilandelayo:
- nge komqondo semithambo ngasiphi komqondo nezinga lokukhula kwengane;
- Alzheimer;
- Parkinson;
- esimweni ukunciphisa inkumbulo nokufunda ikhono, okuhlushwa kahle;
- ene-cerebral palsy;
- ngemva ukulimala nemivimbo, okuholela umgogodla syndrome spastic;
- nge paraplegia, yi-multiple sclerosis.
"Memantine": yokusetshenziswa
Inani, ukubuyekezwa, analogs yalesi izidakamizwa ozijwayele noma ubani emkhayeni abe nesineke komqondo noma nezinye izifo ezihlobene zobuchopho. Regimen kulokhu ukukhetha udokotela. Kodwa imikhaya futhi kudingeka itadishe izidakamizwa "Memantine" imfundo manual. Izidakamizwa analogue futhi wamukela yena kanje:
- amaphilisi ukuphuza ngezikhathi zokudla, ngaphandle ukuhlafuna amanzi amaningi;
- sesondlo yokwelapha eyanele ukuthatha 1-2 amaphilisi ngosuku;
- udinga ukuqala ukwelashwa nge-tablet nengxenye ngosuku, kancane kancane umthamo;
- iziguli abaneminyaka engama 65 Kunconywa ukuba kuthathe ngaphezu 2 amaphilisi ngosuku;
- ukwelashwa lehla "Memantine" inikezwa ngamunye: e ngesonto lokuqala 5 mg ngelanga lesibili - 10 mg, wesithathu - 15-20 mg;
- Isikali ezinconywe udokotela amaconsi zingandiswa kuya ku-30 mg ngosuku, futhi spastic syndrome - ngisho-60 mg;
- izingane ngemva konyaka wonke ukusetshenziswa kwezidakamizwa kungenzeka kuphela amathonsi, umthamo okuyinto kunqunywa ngamunye, ngokuvamile ngesilinganiso 0.5 mg ngayinye kg esisindo ngosuku.
Izimo ukwelashwa
Noma yimuphi Analogue "Memantine" amaphilisi eliqukethe ketshezi asebenzayo esifanayo, akunconyelwe iziguli ezingaphansi kuka engu-18. Akwanele ukufunda umphumela le mithi ebuchosheni ngalesi yobudala.
Contraindicated ekwelapheni noma yiluphi uhlobo lomuthi e azalwa naso galactose ukungabekezelelani, kahle-glucose eyanele phakathi nokukhulelwa kanye lactation. izingxenye isici esiyingqayizivele zomuthi kanye nesenzakalo komzimba nezinto nakho kungaba isithiyo yokwelapha ezinjalo.
Kufanele kuthathwe izinyathelo "Memantine" futhi analogs yayo pathologies nezinso isibindi. Ngemva nokuqedwa metabolites isakhi esiyinhloko esebenzayo, okuyinto akhiwa kwesibindi kwenzeka nge nezinso. Kunconywa ukuthi ukwelashwa Kulezi zimo ngaphansi kokuqondisa kukadokotela futhi umthamo kungenziwa aba nguhhafu. Kuyinto efiselekayo hhayi yokunika leli ukwelashwa iziguli isithuthwane, umfutho wegazi ophakeme, ukuhluleka kwenhliziyo futhi i-hyperthyroidism Ukudlikizela omsakazo engaziwa.
imiphumela emibi izidakamizwa
Lokhu ukulungiselela sina itholakala kuphela kadokotela. Isetshenziswa ngephutha, noma ukuzilimaza yokwelapha, kungabangela imiphumela emibi ukuze isiguli. Ngakho-ke, ngisho nangemva udokotela liyadingeka ukuba isifundo lesi sidakamizwa "Memantine" imfundo manual. Izibuyekezo uqaphele okuvela ezifana side effects:
- isiyezi, labyrinthine syndrome, Gait ukuhlupheka;
- ikhanda, umuzwa wobukhulu ekhanda ;
- ubuthakathaka, ukukhathala;
- ukuquleka, okuvela kuyo zesifo sokuwa;
- ukucindezeleka, ukucasuka, ukusangana;
- isimo ujabule, ukuqwasha;
- isicanucanu, ukuhlanza, kahle wamathumbu umsebenzi, ubuhlungu besisu;
- iyehla iyenyuka wegazi, ukuhluleka kwenhliziyo;
- occlusion semithambo;
- cystitis kanye nezinye izifo kohlelo genitourinary;
- engenhla zokuphefumula ipheshana ukugula, iphika;
- ezifweni ukuba izifo ezibangelwa amagciwane kanye fungal.
imiyalelo okubalulekile ukusetshenziswa kwezidakamizwa
Cishe akukho muntu ku ngokusuka kuyo siqu ukhethe ukuba aphathe 'Memantine ". Yokusetshenziswa, intengo, ukubuyekezwa, analogue ngakho - konke lokhu ikakhulukazi eyaziwa kuphela odokotela. Ngakho-ke, ukuqashwa kukaNksz ukwelashwa okunjalo kubalulekile ukuthola zonke izici isicelo.
- Imithamo kufanele landa kancane kancane, kanye ngesonto.
- Uma degree lesiguli kokuqala zokugula, lapho uyaqhubeka esebenza phakathi ukwelashwa kudingeka uyeke ukushayela nezinye izindlela eziyinkimbinkimbi. Phela, noma iyiphi analog we "Memantine" kungabangela lube buthaka okuhlushwa Ukuwohloka ukuphendula.
- Kubalulekile kakhulu cabanga izidakamizwa ekuhlanganyeleni, ngoba le mithi akuhlangani nezinye izidakamizwa. Abakwazi potentiate "Levodopa" futhi Dopamine yokwamukela abantu abamelene nani, barbiturates, futhi kwehlise umphumela neuroleptics.
- Ayikwazi ukusetshenziselwa "Memantine" futhi analogs yayo "Ketamine", "phenytoin", "amantadine" "quinidine". Lokhu kungayandisa imiphumela anobuthi izidakamizwa. Liphinde sinqatshiwe isifiso sokuba ngibheme ngesikhathi yokwelapha, ngoba kwandisa izinga nicotine egazini.
- Ayikwazi ngokuzimela idlule umthamo watusa yimuphi umuthi udokotela wakho. Kulokhu, aba maningi amathuba okuba ukuthi side effects ukuthuthukisa.
- Ngenxa yezinguquko Ukudla noma ukufakwa kwesicelo antacids kungaluqinisa kakhulu ukubambezela yonke excretion of metabolites "Memantine" kusuka emzimbeni.
"Memantine": nozakwabo
Intengo yale mikhiqizo luyehluka kuye umthamo kanye imikhiqizo yenkampani ruble 400 kuya 2500. Kukhona isifaniso, "Memantine" we ketshezi esebenzayo. Lokhu "Alzeym", "Memantal", "Memaneyrin", "Memantine uhlu lwezincwadi zeBhayibheli", "Memikar", "Memorel", "Noodzheron". Sinenkosi bohlu efanayo isinyathelo futhi iqoqo contra-izinkomba. Amalungiselelo kungahluka khona izingxenye ezengeziwe noma emakamu we ketshezi esebenzayo eyinhloko. Ngenxa yalokhu, i-kahle kungaba ezahlukene ngoba izidakamizwa ezahlukene. Ngakho-ke, isinqumo mayelana nokuthi uluphi uhlobo Analogue "Memantine" ukukhetha for ukwelashwa esimweni ngasinye kumelwe athathe udokotela.
Izibuyekezo sokulungiselela
On ukuphumelela ukwelashwa futhi ohlangothini kungenzeka imiphumela emuthini kuvimbela elikulesi sahluko elithi "Memantine" imfundo manual. Inani analogue kwenza kube kwande. Kodwa odokotela baxwayisa ngokuthi bangase kuphumelele. Yiqiniso, imithi kufanele isikhathi eside. Futhi "Memantine" woqobo owenzwe eJalimane kubiza ruble 1600 ngayinye amaphilisi 30. Analogs yalo, ekhiqizwa eRussia, njengokuthi "Memikar" noma "Memorel" eshibhile, kodwa kungenzeka ehlukile ziqondakala umzimba. Ngakho-ke, ukukhetha imithi kufanele babonane nodokotela. Kodwa ezimweni eziningi ukuthi "Memantine" futhi analogue yayo okubuyayo. Iziguli nezihlobo zabo ziye zaphawula ukuba ngcono okukhulu, ukusebenza kwezimali kanye isimo, ukulahlekelwa kwemisipha izinhlungu zibe nekhanda.
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